ARC 239 is a Selective α2B/2C Adrenoceptor Antagonist
ARC 239 is a selective α2B/2C adrenoceptor antagonist. Besides, ARC 239 binds to CHO cell membranes expressing human recombinant α2A-, α2B- or α2C-adrenoceptor subtypes. α2 adrenoceptor is a G protein-coupled…