![](https://www.Immune-System-Research.com/"wp-content/uploads"/2022/06/Darapladib-is-An-PLA2-Inhibitor-2022-0618.jpg)
Darapladib (SB-480848) is a potent, selective, freely reversible, non-covalently bound, orally active inhibitor of Lp-PLA2 with an IC50 of 0.25 nM, and…
![](https://www.Immune-System-Research.com/"wp-content/uploads"/2022/04/RITANSERIN-2022-0419.png)
α1 Adrenergic receptor is a G protein-coupled receptor (GPCR) associated with GQ heterotrimeric G protein. Besides, α1-adrenergic receptors are including three…
![](https://www.Immune-System-Research.com/"wp-content/uploads"/2022/03/Sulprostone-is-a-Selective-EP3-Receptor-Agonist-2022-03-04-1600x914.png)
Sulprostone (SHB 286), a potent PGE2 analogue, is one of the first EP3 selective agonists. While the half-life of PGE2…
![](https://www.Immune-System-Research.com/"wp-content/uploads"/2021/11/Ro-31-8220-is-a-potent-PKC-Inhibitor-2021-11-18.jpg)
PKC (Protein kinase C) is a family of protein kinase enzymes. In mammals, the PKC family members has four structurally…
![](https://www.Immune-System-Research.com/"wp-content/uploads"/2021/09/BAPTA-AM-a-Ca-2-Chelator-Inhibits-hERG-Channel-2021-10-01.jpg)
Potassium channel, an ion channel, can be found in virtually all species, except for some parasites. Potassium channels have transmembrane…