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Immune System Research

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SARS SARS-CoV SARS-CoV-2

SIMR3030 is a Potent SARS-CoV-2 PLpro Inhibitor for COVID-19 Research

Edward Jenner 2023-06-23

Severe acute respiratory syndrome coronavirus 2 (SARS‑CoV‑2) is a strain of coronavirus that causes COVID-19 (coronavirus disease 2019), the respiratory illness responsible for the COVID-19 pandemic. Although different small-molecule therapeutics…

HIV SARS-CoV

Nirmatrelvir (PF-07321332) is an Orally Active SARS-CoV 3CLpro Inhibitor for COVID-19 Research

Edward Jenner 2023-06-19

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is the cause of the COVID-19 pandemic. Firstly, the coronavirus 3-chymotrypsin-like protease (3CLpro) can control virus replication. Secondly, 3CLpro is responsible for cleaving…

Inflammatory SARS SARS-CoV SARS-CoV-2

Leupeptin is a Broad-Spectrum, Membrane-Permeable Protease Inhibitor

Edward Jenner 2023-04-13

Coronavirus disease 2019 (COVID-19) has caused a huge threat to global public health. Moreover, the constant emergence of variants of concern (VOCs) of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2)…

Coronavirus SARS-CoV SARS-CoV-2

RAY1216 is an Orally Active SARS-CoV-2 Main Protease Slow-tight Inhibitor

Edward Jenner 2023-03-30

As we all know, the SARS-CoV-1 virus caused the 2002-2004 SARS outbreak. Today, we will introduce a virus -- SARS-CoV-2.  SARS-CoV-2 is related to the SARS-CoV-1 virus. SARS-CoV-2 belongs to…

Inflammation migraine Neurological Disease SARS-CoV-2 Viral Immunology

Vazegepant is the First Intranasal CGRP Receptor Antagonist for Migraine

Edward Jenner 2023-03-29

Calcitonin gene-related peptide (CGRP) is a member of the calcitonin peptide family. CGRP has two main forms (α And β). Specifically, CGRP is a highly effective vasodilator. It is important…

Airway Inflammation Infection

Molnupiravir has Antiviral Activity Against Influenza Virus and Multiple Coronaviruses

Edward Jenner 2023-02-28

Coronavirus disease 2019 (COVID-19) is an infectious disease caused by severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2). Symptoms typically include fever, cough, headache, fatigue, difficulty breathing, and loss of smell…

Infection SARS-CoV-2

Beludavimab is a Monoclonal Antibody Targeting SARS-CoV-2 Spike Glycoprotein

Edward Jenner 2023-02-03

SARS‑CoV‑2 (Severe acute respiratory syndrome coronavirus 2) is a strain of coronavirus. However, SARS‑CoV‑2 has caused on going COVID-19 (coronavirus disease 2019) pandemic and led to a serious threat to…

SARS-CoV-2

LY1 is a Selective and Covalent Inhibitor Against SARS-CoV-2 PLpro and Mpro

Edward Jenner 2023-01-30

SARS-CoV-2 PLpro (SARS-CoV-2 papain-like protease) is the largest of the SARS-CoV-2 non-structural proteins (212 kDa). Importantly, the amino acid sequence of SARS-CoV-2PLpro is 98 % identical to related proteases from bat coronaviruses BANAL-52…

Antibodydrug Infection SARS-CoV-2

Masavibart (ZRC3308-A7) is an Anti-SARS-CoV-2 IgG1 Monoclonal Antibody

Edward Jenner 2023-01-06

SARS-COV-2 is a positive-sense single-stranded RNA coronavirus. This virus can cause severe acute respiratory syndrome and spreads between people through aerosols and respiratory droplets. It broke out in early 2020,…

SARS-CoV SARS-CoV-2 Viral Immunology

Bofutrelvir (FB2001) is a SARS-CoV-2 Inhibitor

Edward Jenner 2022-12-27

SARS-CoV-2 is a positive-sense single-stranded RNA coronavirus. This virus can cause severe acute respiratory syndrome and spreads between people through aerosols and respiratory droplets. It broke out in early 2020,…

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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