Irdabisant (CEP-26401) is an Orally Active and BBB Penetrant H3 Receptor Antagonist/Inverse Agonist
Histamine receptors are a type of G protein-coupled receptor (GPCR), including four subtypes: H1, H2, H3, and H4 receptors. They have different functions. For example, the H1 receptor regulates circadian…