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Immune System Research
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Tag: IL-1β

GDC-2394 is an Orally Active and Selective NLRP3 Inhibitor

2022-11-24 Edward Jenner

Nucleotide oligomerization domain (NOD)-like receptors (NLRs) are critical cytoplasmic pattern-recognition receptors (PRRs) that play an important role in the host’s…

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Posted in: Immunology, Innate Immune Filed under: Anti-inflammatory Effect, IL-18, IL-1β, NLRP3

OXSI-2 is an Oxindole Syk Inhibitor

2022-02-25 Edward Jenner

Spleen tyrosine kinase (Syk) is a 72 kDa non-receptor tyrosine kinase. Specifically, Syk is activated by binding the tandem SH2…

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Posted in: Inflammation Filed under: Caspase, IL-1β, Inflammasome, Pyroptosis, ROS

CU-115 is a Selective TLR8 Antagonist

2021-02-03 Edward Jenner

Nucleic acid (NA) sensors are part of the innate immune system. they can recognize multiple forms of intracellular self and…

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Posted in: Inflammation Filed under: IFN, IL-1β, TLR8, TNF-α

DPTIP is a Brain Penetrant N-SMase 2 and Exosome Inhibitor

2020-09-12 Edward Jenner

Neutral sphingomyelinase 2 (nSMase2) catalyzes the formation and release of extracellular vesicles (EVs) . Human nSMase2 catalyzes the hydrolysis of…

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Posted in: Inflammation Filed under: Exosome, IL-1β, N-SMase

JC-171 is a Selective NLRP3 Inflammasome Inhibitor

2020-08-05 Edward Jenner

Multiple sclerosis (MS) is an immune-mediated neurodegenerative disease of the central nervous system (CNS) and is a leading cause of…

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Posted in: Autoimmune Encephalomyelitis Filed under: EAE, IL-1β, Inflammasome, NLRP3

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