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Tag: IL-17

Secukinumab (AIN457) is a Human Monoclonal Antibody Targeted against IL-17A

2021-06-26 Edward Jenner

Interleukin-17 family (IL-17 family) is a pro-inflammatory cystine node cytokine family. After binding to the receptor, IL-17 can activate several…

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Posted in: Immunology, Inflammation, Psoriasis, Skin Inflammation Filed under: IgG1κ, IL-17, IL-17a

BIO-1211 is a Highly Selective and Orally Active α4β1 (VLA-4) Inhibitor

2020-08-27 Edward Jenner

Very Late Antigen-4 (VLA4 or CD49d/CD29) is aα4β1 integrin with a pivotal role in controlling immune cell migration into inflamed…

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Posted in: Autoimmune Disorders, Encephalomyelitis, Inflammation Filed under: EAE, Encephalomyelitis, IFN-γ, IL-17, Integrin, TNF-α, VLA-4, α4β1

BMS-986251 is an Orally Active and Selective RORγt Inverse Agonist

2020-07-07 Edward Jenner

Retinoic acid-related orphan receptor γt (RORγt) is a nuclear hormone receptor (NHR) and belongs to the RORγ family. It exists…

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Posted in: Autoimmune Disorders, Inflammation, Skin Inflammation Filed under: Acanthosis, IL-17, RORγ

SR0987 is a RORγt Agonist to Enhance Protective Immunity

2019-08-31 Edward Jenner

The transcriptional activity of most nuclear receptors (NRs) can be modulated by small lipophilic molecules such as hormones, vitamins, steroids,…

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Posted in: Immunology Filed under: IL-17, Interleukin, PD-1, Th17

SR2211 is a Selective RORγ Inverse Agonist

2019-08-29 Edward Jenner

Retinoic acid receptor-related orphan receptors (RORs) are ligand-dependent transcriptional factors and members of the nuclear receptor superfamily. In fact, RORs…

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Posted in: Autoimmune Disorders, Multiple Sclerosis, Rheumatoid Arthritis Filed under: IL-17, Interleukin, Th17

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