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Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Edward Jenner 2023-09-28

Oxidative stress describes an imbalance between reactive oxygen species (ROS) synthesis and antioxidants. Normally, cells possess antioxidant defense systems that include ROS degrading molecules (ROS scavengers), such as uric acid,…

Inflammatory

Baricitinib is an Orally Active JAK1/2 Inhibitor for Inflammation Research

Edward Jenner 2023-07-20

Janus kinase (JAK) is a family of intracellular, non-receptor tyrosine kinases that transduce cytokine-mediated signals via the JAK-STAT pathway. Importantly, JAK1 and JAK2 are one of the human tyrosine kinase…

Inflammation

KWCN-41 is a Selective RIPK1 Inhibitor for Inflammatory Disorders Research

Edward Jenner 2023-06-14

Necroptosis is a classical mode of cell death co-regulated by RIPK1, RIPK3, and mixed lineage kinase domain-like pseudokinase (MLKL). Necroptosis begins with the activation of death receptors, such as tumor…

Chronic endemic diseases Inflammation

BW 755C is a 5-LO Inhibitor for Inflammation Research

Edward Jenner 2023-06-06

There are only two cyclooxygenases (COX-1 and COX-2) in man, and there are no fewer than 6 lipoxygenases, one of which has been unequivocally linked to human disease, viz., 5-lipoxygenase…

Fungal Fungal Inflammation

Seselin is an Orally Active Antifungal Agent for Inflammation Research

Edward Jenner 2023-06-05

Antifungal agents are drugs that selectively eliminate fungal pathogens from the host with minimal toxicity. Meanwhile, bacteria are prokaryotes and therefore provide many structural and metabolic targets that differ from…

Inflammation

Efipladib is an Orally Active cPLA2α Inhibitor for Inflammation Research

Edward Jenner 2023-05-30

cPLA2α is an intracellular calcium dependent PLA2. It is expressed in a wide variety of tissues and cells. Firstly, cPLA2α can catalyze the release of arachidonic acid (AA) from phospholipids…

Auto-Inflammatory Inflammation

BI 1015550 is an Orally Active PDE4B Inhibitor for Inflammation Research

Edward Jenner 2023-04-27

PDE4B is an enzyme that in humans is encoded by the PDE4B gene. Importantly, PDE4B is involved in dopamine-associated and stress-related behaviors. Particularly, study show that reduction in PDE4B activity…

Autoimmune diseases Inflammatory Uncategorized

SRTCX1003 is an Orally Active SIRT1 Activator for Inflammatory Research

Edward Jenner 2023-04-19

Sirtuin (Sir2 proteins) is a class of proteins. And it possesses either mono-ADP-ribosyltransferase, or deacylase activity, including deacetylase, desuccinylase, demalonylase, demyristoylase and depalmitoylase activity. Sirtuins regulate important biological pathways in…

Infection Inflammation

Eritoran is a TLR4 Antagonist for Influenza Virus Infection Research.

Edward Jenner 2023-04-18

TLR4 is a transmembrane protein that belongs to the toll-like receptor family member of the pattern recognition receptor (PRR) family. Firstly, activation of Toll-like receptor 4 (TLR4) promotes the intracellular…

Inflammation migraine Neurological Disease SARS-CoV-2 Viral Immunology

Vazegepant is the First Intranasal CGRP Receptor Antagonist for Migraine

Edward Jenner 2023-03-29

Calcitonin gene-related peptide (CGRP) is a member of the calcitonin peptide family. CGRP has two main forms (α And β). Specifically, CGRP is a highly effective vasodilator. It is important…

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Recent Posts

  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
  • Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research
  • Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research
  • Doravirine is a HIV-1 Inhibitor for Infection Research

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

Up to date immunology information

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