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Inflammation

SSK1, a β-Galactosidase-targeted Prodrug, Attenuates Inflammation

Edward Jenner 2021-07-22

β-Galactosidase, a glycoside hydrolase family, catalyzes the cleavage of glycosidic bonds β-Galactoside is hydrolyzed to monosaccharide. Specifically, β-Galactosidase is a kind of exoglycosidase, which can hydrolyze the protein formed between…

Arthritis Inflammation Psoriasis

BMS-582949 is an Orally Active p38α MAPK Inhibitor

Edward Jenner 2019-08-23

BMS-582949 was identified as a highly selective p38α MAP kinase inhibitor as early in 2010. Moreover, it has entered into clinical trials for further development and clinical studies in inflammatory…

Endometriosis Fibrosis Inflammation Pulmonary Fibrosis

FR 167653, an Orally Active p38 MAPK Inhibitor, Inhibits Cytokine Production

Edward Jenner 2019-08-05

Various types of cytokinesuchemokines react with their receptors. They transduce extracellular signals into intracellular response through a mitogen-activated protein kinase (MAPK) signalling cascade. Furthermore, p38 MAPK signalling might play an…

Inflammation

MW-150, an Orally Active p38α MAPK Inhibitor, Modulates Cytokine Production and Cognitive Outcomes

Edward Jenner 2019-08-04

Currently, a void exists for serine/threonine protein kinase inhibitor drugs and central nervous system indications. Stress kinases are of special interest in neurological and neuropsychiatric disorders, because of their involvement…

Arthritis Rheumatoid Arthritis

SD 0006 is an Orally Active MAPK p38α Inhibitor for the Treatment of Rheumatoid Arthritis

Edward Jenner 2019-08-02

In previous blogs, we have introduced a few MAPK p38 inhibitors. As a result, MAPK p38 plays an important role in many diseases, including cancer and inflammatory diseases. Today, I’d…

Arthritis Inflammation

AL 8697 is an Orally Active and Specific p38α MAPK Inhibitor

Edward Jenner 2019-07-17

A wide range of cellular stresses can activate mammalian p38 MAPKs, or it is in response to inflammatory cytokines. The p38 MAPK subfamily can further be divided into two distinct…

Asthma

SB 239063 is a Potent p38 MAPK Inhibitor for Treatment of Asthma

Edward Jenner 2019-07-07

Asthma is a chronic inflammatory disease of the lungs. It is a common disease due to genetic and environmental factors. However, there is no cure for this disease. We can…

Arthritis Rheumatoid Arthritis

Doramapimod is a Highly Potent p38 MAPK Inhibitor with Anti-inflammatory Acitivity

Edward Jenner 2019-06-15

The mitogen-activated protein kinase (MAPK) p38a is activated by environmental stimuli, bacterial products and cytokines. It plays a critical role in the production of proinflammatory cytokines such as TNF-a and…

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  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
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  • Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research
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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

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