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Tag: PDE4

LEO 39652 is a Dual-Soft PDE4 Inhibitor

2021-03-18 Edward Jenner

Atopic dermatitis (AD) is a chronic inflammatory skin disease. the characterizes of AD are eczematous lesions and intense itching. The…

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Posted in: Atopic Dermatitis, Skin Inflammation Filed under: PDE4

MR-L2 is a Reversible and Noncompetitive Allosteric Activator of Long-Isoform PDE4

2020-12-19 Edward Jenner

Cyclic AMP (cAMP) is a universal second messenger in cells of all biological systems. Specifically, cAMP homeostasis is affected by…

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Posted in: Neuroimmunology Filed under: cAMP, PDE4, PDE4D5, UCR1

GSK356278 is a Selective and Orally Bioavailable PDE4 Inhibitor

2020-10-21 Edward Jenner

Phosphodiesterase-4 (PDE4) acts as an intracellular non-receptor enzyme that modulates inflammation and epithelial integrity. GSK356278, a potent, selective, brain-penetrant phosphodiesterase…

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Posted in: Inflammation Filed under: Anxiolytic, PDE4, TNF-α

FCPR03 is a Selective Phosphodiesterase 4 (PDE4) Inhibitor

2020-07-21 Edward Jenner

Phosphodiesterase 4 (PDE4) is an enzyme mainly expresses in the central nervous system, smooth muscle, cardiovascular.  In neuronal cells, PDE4…

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Posted in: Inflammation Filed under: Antidepressant, PDE4

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