Skip to content
Immune System Research
Up to date immunology information.

Tag: RIPK

GSK481 is a Mono-Selective RIP1 Kinase Inhibitor

2019-09-09 Edward Jenner

Recent research shows that RIP1 kinase activity is an important driver of TNF-mediated inflammation and pathology. Genetic evidence of mice…

Continue Reading →

Posted in: Inflammation Filed under: RIPK, TNF

GSK583 is an Orally Active and Selective RIP2 Kinase Inhibitor

2019-09-02 Edward Jenner

In previous blogs, I have introduces several RIPK inhibitors, including RIP1 inhibitors RIPA-56, PK68, GSK547, GNE684, and GSK2982772. But the…

Continue Reading →

Posted in: Inflammation Filed under: NOD1, NOD2, RIPK

GSK2983559 is a Specific and Oral Active RIP2 Kinase Inhibitor for Inflammatory Diseases

2019-09-01 Edward Jenner

The innate immune system is a key driver of our immune response from birth. It provides an immediate response to…

Continue Reading →

Posted in: Auto-Inflammatory Filed under: Anti-Inflammatory, RIPK

RIPA-56 is a Selective RIP1 Inhibitor for the Treatment of SIRS

2019-08-27 Edward Jenner

Necrosis is the death of cells and tissues. The kinase activity of receptor-interacting protein kinase 1 (RIP1/RIPK1) and/or RIP3/RIPK3 mediates…

Continue Reading →

Posted in: Systemic Inflammatory Response Syndrome Filed under: Apoptosis, Necroptosis, RIPK, SIRS, TNF

PK68, a type II Inhibitor of RIPK1, Has potential to Treat Inflammatory Disorders and Cancer Metastasis

2019-07-28 Edward Jenner

Necroptosis is a form of regulated necrosis controlled by receptor-interacting kinase 1 (RIPK1), RIPK3, and mixed lineage kinase domain-like protein…

Continue Reading →

Posted in: Cancer Immunology, Colitis, Inflammation Filed under: Metastasis, RIPK

Post navigation

Page 1 of 2
1 2 Next →
Loading

Archives

Recent Posts

  • Beludavimab is a Monoclonal Antibody Targeting SARS-CoV-2 Spike Glycoprotein 2023-02-03
  • Tibulizumab (LY 3090106) is a Tetravalent Bispecific mAb Targeting BAFF and IL-17A 2023-01-31
  • LY1 is a Selective and Covalent Inhibitor Against SARS-CoV-2 PLpro and Mpro 2023-01-30

Categories

  • Abdominal Aortic Aneurysm
  • Acanthosis
  • Achondroplasia
  • Acute Pancreatitis
  • Acute Radiation Syndrome
  • AIDs
  • Airway Immunology
  • Airway Inflammation
  • Allergy
  • Alzheimer
  • Analgesia
  • Antibodydrug
  • Antigen-Induced Arthritis
  • Arterial Thrombosis
  • Arthritis
  • Asthma
  • Atherosclerosis
  • Atopic Dermatitis
  • Atopic Dermatitis
  • Atrial Fibrillation
  • Autism
  • Auto-Inflammatory
  • Autoimmune Disorders
  • Autoimmune Encephalitis
  • Autoimmune Encephalomyelitis
  • Bacterial
  • Bronchial Airway Infection
  • Cancer Immunology
  • Cancer Immunotherapy
  • Cardiovascular
  • Chemokines
  • Chronic Arthritis
  • Chronic Heart Failure
  • Chronic Hepatitis B
  • Chronic Obstructive Pulmonary Disease
  • Chronic Obstructive Pulmonary Disease
  • Chronic Urticaria
  • Cognitive Disorders
  • Colitis
  • Collagen-Induced Arthritis
  • Complement System
  • Crohn's Disease
  • Degenerative disease
  • Diabetic Complication
  • DNV
  • Dye
  • EMCV
  • Encephalomyelitis
  • Encephalomyelitis
  • Endocrinology
  • Endometriosis
  • Enterovirus
  • Epilepsy
  • Fabry Disease
  • Fibrosis
  • FIPV
  • Fungal
  • Fungal
  • Growth & Development
  • Haemophilia
  • HBV
  • HCV
  • Hemorrhagic Disorder
  • Hepatic steatosis
  • Hepatic steatosis
  • Hepatitis
  • Hepatitis
  • Hepatitis C Virus
  • Hereditary Angioedema
  • HIV
  • Homeostasis
  • HPV
  • HSV
  • hypertension
  • Idiopathic Pulmonary Fibrosis
  • Immune Checkpoint
  • Immune homeostasis
  • Immune Rejection
  • Immunodeficiency
  • Immunology
  • Immunotherapy
  • Infection
  • Inflammation
  • Influenza Virus
  • Innate Immune
  • Intestinal Inflammation
  • Ischemic stroke
  • Kidney Fibrosis
  • Kidney immune
  • Kidney Injury
  • Lower Respiratory Infection
  • Lung Inflammation
  • Lupus Nephritis
  • Malaria
  • Mesothelioma
  • Metabolic Disease
  • Metabolic Disorder
  • Multiple Sclerosis
  • Multiple Sclerosis
  • Neuroimmunology
  • Neurological Disease
  • obesity
  • Osteoarthritis
  • Osteoporosis
  • Pancreatitis
  • Pancreatitis
  • Parasite
  • Parasite
  • Parkinson’s
  • Periodontitis
  • Peritonitis
  • Psoriasis
  • Psoriasis
  • Pulmonary Arterial Hypertension (PAH)
  • Pulmonary Fibrosis
  • RABV
  • RABV
  • Renal Fibrosis
  • Respiratory Infection
  • Retinal Vascular Diseases
  • Rheumatoid Arthritis
  • Rheumatoid Arthritis
  • Rhinitis
  • Rhinovirus
  • SARS
  • SARS-CoV
  • SARS-CoV-2
  • Schizophrenia
  • Seizure
  • Sepsis
  • Skin Inflammation
  • Stroke
  • Systemic Inflammatory Response Syndrome
  • Systemic Lupus Erythematosus
  • Systemic Scleroderma
  • Thrombosis
  • Tuberculosis
  • Type 2 Diabetes Mellitus
  • Ulcerative Colitis
  • Uncategorized
  • Updated
  • Venous Ulcers
  • Viral Immunology

Tags

5-HT Anti-Inflammatory Anti-Tumor Antibacterial Antibiotic Antifungal Antimalarial Antitumor Antiviral Apoptosis Autophagy Breast Cancer Chemokines COPD COVID-19 Cytokine Diabetes Dopamine EGFR HBV HCV HIV IL-1β IL-6 Infection Inflammasome Integrin Interferon Interleukin IPF Leukemia Low Toxicity Monoclonal Antibody Multidrug Resistance NF-κB p38 MAPK Proteasome ROS SARS-CoV SARS-CoV-2 T Cell Th17 TLR TNF TNF-α
Copyright © 2023 Immune System Research — Primer WordPress theme by GoDaddy