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Tag: NF-κB

CMC2.24 is an Orally Active Tricarbonylmethane Agent

2021-01-27 Edward Jenner

RAS is the name of a series of related proteins commonly expressed in all cell lineages and organs. Specifically, RAS…

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Posted in: Osteoarthritis Filed under: HIF-2α, MMP, NF-κB, RAS

TML-6 Inhibits the Synthesis of the β-amyloid Precursor Protein and β-amyloid

2021-01-12 Edward Jenner

Amyloid beta (Aβ) is a major component of amyloid plaques found in the brains of patients with Alzheimer’s disease. Specifically,…

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Posted in: Alzheimer Filed under: Amyloid, mTOR, NF-κB, Nrf2

SP-100030 is a Potent NF-κB and Activator Protein-1 (AP-1) Inhibitor

2020-10-01 Edward Jenner

Nuclear factor-κB (NF-κB) represents a family of inducible transcription factors. The transcription factor NF-κB regulates multiple aspects of innate and…

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Posted in: Arthritis, Collagen-Induced Arthritis, Inflammation Filed under: AP-1, Interleukin, Jurkat, NF-κB, TNF-α

GS143 is a Selec­tive IκBα Ubiquitination Inhibitor

2020-09-01 Edward Jenner

GS143 is a selective IκBα ubiquitination inhibitor with an IC50 of 5.2 μM for SCFβTrCP1-mediated IκBα ubiquitylation. Firstly, when GS143…

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Posted in: Asthma, Bronchial Airway Infection, Cancer Immunology, Inflammation Filed under: IκB, NF-κB, p53, Th2, Ubiquitination, β-catenin

MS417 is a BET-Specific BRD4 Inhibitor

2020-01-17 Edward Jenner

NF-κB-mediated inflammation is a major pathology in kidney diseases, such as non-kidney inflammatory diseases, and rheumatoid arthritis. HIV infection in…

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Posted in: HIV, Inflammation, Rheumatoid Arthritis, Viral Immunology Filed under: BRD4, HIV, HIVAN, NF-κB

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