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Category: Cancer Immunology

WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis

2021-02-25 Edward Jenner

Much of the past effort has focused on targeting caspases, proteases that mediate many of the hallmarks of apoptotic cell…

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Posted in: Cancer Immunology Filed under: Apoptosis, BAK, VDAC2

SBP-7455 is an Orally Active Dual ULK1/ULK2 Autophagy Inhibitor

2021-01-22 Edward Jenner

Autophagy is a multi-step pathway initiated through the ULK preinitiation complex, which consists of unc-51-like autophagy activating kinase 1 (ULK1)…

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Posted in: Cancer Immunology Filed under: Autophagy, Breast Cancer, TNBC, ULK

KMH-233 is a Reversible and Selective LAT1 Inhibitor

2021-01-18 Edward Jenner

Amino acids are essential for protein synthesis, they are supporting cell growth, and metabolism. System L belongs to the family…

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Posted in: Cancer Immunology Filed under: Anti-proliferative, Anti-Tumor, Breast Cancer, LAT1

Osimertinib is an Irreversible and Mutant Selective EGFR Inhibitor

2021-01-13 Edward Jenner

Epidermal growth factor receptor (EGFR) is a transmembrane receptor tyrosine kinase protein. EGFR plays an important role in controlling cell…

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Posted in: Cancer Immunology, Cancer Immunotherapy Filed under: EGFR, IGF1R, T790M

CB-5083 is a Selective and Orally Bioavailable p97 Inhibitor

2020-12-17 Edward Jenner

The AAA+ ATPase p97 is essential to a wide range of cellular functions. The p97 acts downstream from ubiquitin signaling…

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Posted in: Cancer Immunology Filed under: Anti-Tumor, Apoptosis, ATPase, Multiple Myeloma, p97, Proteasome, TPD

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Recent Posts

  • Enpatoran is an Orally Active and Dual TLR7/8 Inhibitor 2021-02-27
  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24

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