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Immune System Research
Up to date immunology information.

Category: Colitis

Glepaglutide (ZP1848) is a potent GLP-2R agonist, good for inflammatory bowel disease (IBD) and Crohn’s disease

2022-11-14 Edward Jenner

Glucagon-like peptide 2 (GLP-2) is an enterotrophic hormone consisting of 33 amino acids. It derives from a glucagon pro-peptide encoded…

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Posted in: Colitis, Crohn's Disease, Intestinal Inflammation Filed under: Crohn's disease, GLP-2, GLP-2R, inflammatory bowel disease

SR12418 is a REV-ERB-specific Synthetic Ligand

2022-10-15 Edward Jenner

REV-ERB is a member of the nuclear receptor superfamily consisting of two similar proteins: REV-ERBα and REV-ERBβ. Like other NRs,…

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Posted in: Autoimmune Disorders, Colitis, Encephalomyelitis, Inflammation Filed under: Circadian Rhythm, Glucose Metabolism, lipid metabolism, Related Orphan Receptors, REV-ERB

NIC-0102 is an Orally Active Proteasome Inhibitor, Specifically Inhibiting NLRP3 Inflammatory Vesicle Activation

2022-10-06 Edward Jenner

Nucleotide oligomerization domain (NOD)-like receptors (NLRs) are critical cytoplasmic pattern-recognition receptors (PRRs). They play an important role in the host\’s…

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Posted in: Colitis, Inflammation, Ulcerative Colitis Filed under: Anti-Inflammatory, NLRP3-ASC, pro-IL-1β, Proteasome, Ulcerative Colitis

XL01126 is a Potent and Fast LRRK2 Degrader for Parkinson’s Disease Research

2022-09-05 Edward Jenner

Leucine Rich Repeat Kinase 2 (LRRK2) is a member of the leucine-rich repeat kinase family. Researchers found that the mutations…

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Posted in: Colitis, Crohn's Disease, Neurological Disease, Parkinson’s Filed under: Crohn's disease, LRRK2, Parkinson's disease

Teprenone, an Anti-ulcer Drug, is an Inducer of Heat Shock Proteins (HSPs)

2022-06-04 Edward Jenner

Ulcer is caused by discontinuity or break in a bodily membrane, which can damage normal function of the affected organ.…

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Posted in: Ulcerative Colitis Filed under: HSPs, Teprenone, Ulcer

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