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Category: Colitis

Teprenone, an Anti-ulcer Drug, is an Inducer of Heat Shock Proteins (HSPs)

2022-06-04 Edward Jenner

Ulcer is caused by discontinuity or break in a bodily membrane, which can damage normal function of the affected organ.…

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Posted in: Ulcerative Colitis Filed under: HSPs, Teprenone, Ulcer

Etrasimod is a Selective and Orally Active S1P1 Receptor Antagonist

2022-04-07 Edward Jenner

Etrasimod is a potent, selective, and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor. And the IC50 value is 1.88 nM in…

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Posted in: Colitis, Rhinitis, Ulcerative Colitis Filed under: Atopic Dermatitis, Crohn Disease, Pyoderma Gangrenosum, S1P1

NX-13 Targets and Activates NLRX1 to Induce Immunometabolic Changes

2021-08-07 Edward Jenner

NLRX1 is a highly conserved nucleotide-binding domain (NBD) and a member of the leucine-rich repeat (LRR) family (NLR). Specifically, NLRX1…

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Posted in: Colitis, Crohn's Disease, Ulcerative Colitis Filed under: NLRX1

BMS-986202 is an Orally Active Tyk2 Inhibitor that Binds to Tyk2 JH2

2021-02-06 Edward Jenner

Tyrosine kinase 2 (Tyk2) is a non-receptor tyrosine kinase belonging to the Janus kinase (JAK) family. Specifically, the mammalian JAK…

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Posted in: Acanthosis, Colitis, Systemic Lupus Erythematosus Filed under: CYP2C19, Tyk2

Plecanatide is an Orally Active Guanylate Cyclase-C (GC-C) Receptor Agonist

2020-09-25 Edward Jenner

Guanylyl cyclase-C (GC-C) is a transmembrane receptor for bacterial heat-stable enterotoxin and the mammalian peptides guanylin and uroguanylin. Guanylyl cyclase-C…

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Posted in: Colitis Filed under: cGMP, GC-C, TNBS

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