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Category: Inflammation

GSK-J4 is a Dual Inhibitor of H3K27me3/me2-Demethylases JMJD3/KDM6B and UTX/KDM6A

2021-02-18 Edward Jenner

H3K27me3 is an epigenetic modification of DNA packaging protein histone H3. Specifically, it is a marker for the trimethylation of…

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Posted in: Autoimmune Disorders, Inflammation Filed under: Apoptosis, ER Stress, H3K27, JMJD3, KDM6A, KDM6B, TNF-α

BMS-986202 is an Orally Active Tyk2 Inhibitor that Binds to Tyk2 JH2

2021-02-06 Edward Jenner

Tyrosine kinase 2 (Tyk2) is a non-receptor tyrosine kinase belonging to the Janus kinase (JAK) family. Specifically, the mammalian JAK…

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Posted in: Acanthosis, Colitis, Systemic Lupus Erythematosus Filed under: CYP2C19, Tyk2

CU-115 is a Selective TLR8 Antagonist

2021-02-03 Edward Jenner

Nucleic acid (NA) sensors are part of the innate immune system. they can recognize multiple forms of intracellular self and…

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Posted in: Inflammation Filed under: IFN, IL-1β, TLR8, TNF-α

BMS 753 is a Selective RARα Agonist

2021-02-02 Edward Jenner

RARs (α,β, and γ and their isoforms) and RXRs (α,β, and γ and their isoforms) are members of the nuclear…

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Posted in: Inflammation Filed under: RARα

LY-311727 is a Secretory non-Pancreatic Phospholipase A2 (sPLA2) Inhibitor

2021-01-28 Edward Jenner

Phospholipase A2 (PLA2s) is an enzyme that cleaves fatty acids in the second position of phospholipids. Specifically, PLA2s can specifically…

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Posted in: Inflammation Filed under: Phospholipase, sPLA2

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  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24
  • FSCPX is a Selective Irreversible Antagonist of A1AR 2021-02-23

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