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Immune System Research
Up to date immunology information.

Category: obesity

GSK837149A is a Selective Human Fatty Acid Synthase (FASN) inhibitor

2023-02-09 Edward Jenner

Fatty acid synthase (FASN) is a central regulator of lipid metabolism. FASN provides the fatty acids needed to sustain tumor…

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Posted in: Cancer Immunology, obesity Filed under: Breast Cancer, fatty acid synthase, GSK837149A, ketoacyl reductase, obesity

Crotedumab (REGN1193) is an Anti-GCGR IgG4 Monoclonal Antibody

2023-01-10 Edward Jenner

Glucagon plays an important role in glucose metabolism. Upon hypoglycemia, pancreatic alpha cells can secrete glucagon which stimulates hepatic glucose…

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Posted in: Antibodydrug, Diabetic Complication, obesity, Type 2 Diabetes Mellitus Filed under: GCGR, Glucose, Type 2 Diabetes

LY3437943 is a Triple Agonist of GCGR/GIPR/GLP-1R

2022-11-10 Edward Jenner

Glucagon receptor (GCGR), a 62 kDa protein, is a member of the class B G-protein coupled family of receptors. GCGR…

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Posted in: Metabolic Disease, obesity, Type 2 Diabetes Mellitus Filed under: anti-obesity, GLP-1, Glucose Metabolism, lipid metabolism

Cotadutide is a Potent GLP-1 and GCGR Dual Agonist

2022-11-05 Edward Jenner

Glucagon-like peptide-1 (GLP-1) is a 30- or 31-amino acid peptide hormone produced and secreted by intestinal enteroendocrine L-cells and certain neurons within the…

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Posted in: Metabolic Disease, obesity, Type 2 Diabetes Mellitus Filed under: Diabetes, GCGR, GLP-1, obesity, T2D

JBSNF-000028 is an Orally Active NNMT Inhibitor, with Anti-obesity Activity

2022-11-01 Edward Jenner

Nicotinamide N-methyltransferase (NNMT) is a metabolic enzyme. Specifically, NNMT is involved in controlling methylation potential and influencing epigenetic modification of…

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Posted in: obesity Filed under: JBSNF-000028, metabolic disorder, nicotinamide N-methyltransferase, NNMT, obesity, orally
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