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Category: HIV

Aplaviroc (AK 602) is a CCR5 Antagonist

2022-05-07 Edward Jenner

Aplaviroc (AK 602), an SDP derivative, is a potent CCR5 antagonist. Additionally, the IC50s  are 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL, and…

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Posted in: HIV, Infection Filed under: CCR5, HIV

Rottlerin is a Specific PKC Inhibitor

2022-01-07 Edward Jenner

Protein kinase C (PKC) is a family of protein kinase enzymes with 15 isoforms that can regulate the protein function.…

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Posted in: HIV, Immunodeficiency, RABV Filed under: Apoptosis, Autophagy, HIV, mTORC, PKC, RABV

Nelfinavir (AG-1341) is an Orally Active HIV-1 Protease Inhibitor

2021-09-25 Edward Jenner

HIV protease is a homodimeric aspartyl protease. It is worth noting that, HIV protease is crucial for the viral life-cycle.…

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Posted in: Cancer Immunology, HIV, SARS-CoV, Viral Immunology Filed under: Anticancer, COVID-19, HIV-1, SARS-CoV, U266

Cobicistat is a Selective CYP3A Inhibitor and a Pharmacokinetic Enhancer of HIV Inhibitors

2020-12-22 Edward Jenner

The highly active antiretroviral therapy (HAART) can transform the human immunodeficiency virus (HIV) infection into a manageable chronic disease in…

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Posted in: HIV, Viral Immunology Filed under: Antiviral, CYP3A, HIV

TC14012 is a Selective CXCR4 Inverse Agonist and CXCR7 Agonist

2020-08-19 Edward Jenner

CXC chemokine receptors are the complete membrane proteins and they can specifically bind and respond to CXC chemokine family cytokines.…

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Posted in: Cancer Immunology, HIV, Viral Immunology Filed under: Antitumor, CCR5, CXCR4, CXCR7

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