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Immune System Research
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Category: Analgesia

SSR504734 is an Orally Active, Selective and Reversible GlyT1 Inhibitor

2022-09-22 Edward Jenner

Glycine transporters (GlyTs) are the Na+/Cl–-dependent plasmalemmal neurotransmitter transporters. GlyTs comprise GlyT1 and GlyT2. They serve to terminate the signaling…

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Posted in: Analgesia, Cognitive Disorders, Epilepsy, Neurological Disease, Schizophrenia Filed under: Anti-anxiety, Anti-depression, Anti-schizophrenia

Flavoxate is a Potent and Competitive PDE inhibitor

2022-08-06 Edward Jenner

Phosphodiesterases (PDEs) are enzymes that catalyze the hydrolysis of the 3′ cyclic phosphate bond of cyclic nucleotides. PDEs can break…

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Posted in: Analgesia, Inflammation Filed under: Overactive Bladder, Urinary Tract Infection

SB-612111 is a Potent Human Opiate Receptor-Like Orphan Receptor (ORL-1) Antagonist

2020-06-10 Edward Jenner

Nociceptin, as a 17-amino acid peptide, is a potent endogenous agonist for the opiate receptor-like orphan receptor (ORL-1). It exhibits…

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Posted in: Analgesia Filed under: GPCR, Opioid, ORL

UNC3230 is a Selective and ATP-Competitive PIP5K1C Inhibitor

2020-06-04 Edward Jenner

Phosphatidylinositol-4-phosphate 5-kinase type-1C (PIP5K1C) is a lipid kinase that regulates focal adhesion dynamics and cell attachment through the site-specific formation…

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Posted in: Analgesia Filed under: Anti-Tumor, PIP5K1C
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