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Category: Immunodeficiency

GS-6207 is a First-In-Class HIV-1 Capsid Inhibitor with Long-Acting Potential

2019-12-04 Edward Jenner

Exceptional developments in combination antiretroviral therapy (cART) have transformed HIV/AIDS from a deadly pandemic to chronic and manageable disease. HIV-1…

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Posted in: HIV, Immunodeficiency, Viral Immunology Filed under: HIV

Identification of a HIV 1 Maturation Inhibitor GSK3532795

2019-05-18 Edward Jenner

Human immunodeficiency virus (HIV) is a threat to humans and a serious issue for public health worldwide. Especially, acquired immune…

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Posted in: AIDs, Immunodeficiency, Viral Immunology Filed under: HIV

MLT-748, an Allosteric MALT1 Inhibitor, is a Molecular Corrector to Rescue Function in Immunedeficiency

2019-05-12 Edward Jenner

In previous blog “MLT-747, an Allosteric MALT1 Inhibitor for Immunodeficiency Research”, we introduced MLT-747 as a potent, selective, allosteric inhibitor…

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Posted in: Immunodeficiency Filed under: MALT

MLT-747, an Allosteric MALT1 Inhibitor for Immunodeficiency Research

2019-05-11 Edward Jenner

Immunodeficiency is a state, in which the immune system’s ability is absent. It is not able to fight against cancer…

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Posted in: Immunodeficiency Filed under: MALT

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Recent Posts

  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24
  • FSCPX is a Selective Irreversible Antagonist of A1AR 2021-02-23

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Anti-Inflammatory Anti-Tumor Antibacterial Antimalarial Antitumor Antiviral Apoptosis Autophagy Breast Cancer Btk Chemokines COPD COX Cytokine EGFR ER Stress HBV HCV HDAC HIV IFN IL-6 IL-17 Infection Integrin Interferon Interleukin Leukemia Low Toxicity Multidrug Resistance Necroptosis NF-κB p38 MAPK PI3K PPI Proteasome RIPK STAT STING T Cell Th17 TLR TNF TNF-α α4β1
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