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Immune System Research
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Category: Epilepsy

PRE-084 is a S1R Agonist for Cardiovascular and Neurological Disease Research

2023-05-24 Edward Jenner

The sigma-1 receptor (σ1R, S1R), one of two sigma receptor subtypes, is a chaperone protein at the endoplasmic reticulum (ER)…

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Posted in: Alzheimer's disease, Cancer, Cardiovascular, Epilepsy, Schizophrenia Filed under: Alzheimer´s Disease, PRE-084, sigma-1 Receptor

LY456236 is an Orally Active mGlu1 Receptor Antagonist for Neurological Disease Research

2023-04-25 Edward Jenner

Epilepsy is one of the most common neurological diseases in the world. Firstly, Epilepsy affects people of all ages, races,…

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Posted in: Epilepsy Filed under: Epilepsy, LY456236, mGlu1, OCCM-30

JNJ-56022486 is an Orally Active Negative AMPA Receptor Modulator for Epilepsy Research

2023-03-07 Edward Jenner

Glutamate is the primary excitatory neurotransmitter in the mammalian brain. AMPA (α-amino-3-hydroxyl-5-methyl-4-isoxazole-propionic acid) is the subtype of glutamate receptors and…

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Posted in: Epilepsy, Neurological Disease Filed under: AMPA, CNS disorders, Epilepsy, JNJ-56022486, TARP-γ8

Fuzapladib (IS-741) is A Potent Phospholipase A2 Inhibitor

2023-02-16 Edward Jenner

Phospholipase is a member of a very complex group of enzymes that break down phospholipids into fatty acids and other…

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Posted in: Alzheimer, Epilepsy, Inflammation, Ischemia, Multiple Sclerosis, Neurological Disease Filed under: IL-8, Inflammation, Neuroinflammation, Neurological disease, PAF, PG, Phospholipase, PLA2

SSR504734 is an Orally Active, Selective and Reversible GlyT1 Inhibitor

2022-09-22 Edward Jenner

Glycine transporters (GlyTs) are the Na+/Cl–-dependent plasmalemmal neurotransmitter transporters. GlyTs comprise GlyT1 and GlyT2. They serve to terminate the signaling…

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Posted in: Analgesia, Cognitive Disorders, Epilepsy, Neurological Disease, Schizophrenia Filed under: Anti-anxiety, Anti-depression, Anti-schizophrenia

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