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Category: Ulcerative Colitis

Teprenone, an Anti-ulcer Drug, is an Inducer of Heat Shock Proteins (HSPs)

2022-06-04 Edward Jenner

Ulcer is caused by discontinuity or break in a bodily membrane, which can damage normal function of the affected organ.…

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Posted in: Ulcerative Colitis Filed under: HSPs, Teprenone, Ulcer

Etrasimod is a Selective and Orally Active S1P1 Receptor Antagonist

2022-04-07 Edward Jenner

Etrasimod is a potent, selective, and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor. And the IC50 value is 1.88 nM in…

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Posted in: Colitis, Rhinitis, Ulcerative Colitis Filed under: Atopic Dermatitis, Crohn Disease, Pyoderma Gangrenosum, S1P1

NX-13 Targets and Activates NLRX1 to Induce Immunometabolic Changes

2021-08-07 Edward Jenner

NLRX1 is a highly conserved nucleotide-binding domain (NBD) and a member of the leucine-rich repeat (LRR) family (NLR). Specifically, NLRX1…

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Posted in: Colitis, Crohn's Disease, Ulcerative Colitis Filed under: NLRX1

BRD5529 is a Selective CARD9–TRIM62 PPI Inhibitor

2019-11-18 Edward Jenner

The allele family CARD9 variant relates to increased or protected risk of inflammatory bowel disease (IBD). Moreover, the susceptible variant…

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Posted in: Colitis, Inflammation, Ulcerative Colitis Filed under: CARD9, TRIM62, Ubiquitination

KAG-308 is an Orally Active EP4-Selective Agonist for Ulcerative Colitis Treatment

2019-07-15 Edward Jenner

As we all know, Colitis is a kind of inflammatory diseases. Sometimes it is acute and long term, makes patients…

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Posted in: Colitis, Ulcerative Colitis Filed under: Anti-Tumor, TNF
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