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Category: Neuroimmunology

PF-06256142 is a Selective and BBB Penetrated Orthosteric Agonist of the D1 Receptor

2021-03-04 Edward Jenner

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the central nervous system (CNS) of vertebrates.…

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Posted in: Neuroimmunology, Neurological Disease Filed under: CNS, Dopamine

YM90K is a Selective AMPA Receptor Antagonist with Neuroprotective Actions

2021-02-20 Edward Jenner

AMPA receptors are ionic transmembrane receptors of glutamate, which mediate rapid synaptic transmission in the central nervous system (CNS). Specifically,…

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Posted in: Neuroimmunology, Neurological Disease Filed under: AMPA, Ischemia

AZD1940 is an Orally Active Cannabinoid CB1/CB2 Receptor Agonist

2021-02-09 Edward Jenner

Cannabinoid receptor is a kind of cell membrane receptor in the G protein-coupled receptor superfamily. Specifically, the cannabinoid receptor contains…

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Posted in: Neuroimmunology, Neurological Disease Filed under: Analgesia, Cannabinoid, CB1, CB2

Lu AE98134 is a Selective Positive Modulator of NaV1.1 Channels

2021-01-30 Edward Jenner

Sodium channels are integral membrane proteins that form ion channels and conduct sodium ions (Na+) through the plasma membrane. These…

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Posted in: Neuroimmunology, Neurological Disease Filed under: NaV1.1, NaV1.6, Schizophrenia

URB937 is a FAAH Inhibitor

2021-01-09 Edward Jenner

Neurotransmitters participate in pain perception effectively. One prominent example of peripheral regulation is provided by the endogenous opioids, which are…

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Posted in: Inflammation, Neuroimmunology Filed under: Anandamide, Drugdiscovery, FAAH

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