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Category: Skin Inflammation

BMS-986202 is an Orally Active Tyk2 Inhibitor that Binds to Tyk2 JH2

2021-02-06 Edward Jenner

Tyrosine kinase 2 (Tyk2) is a non-receptor tyrosine kinase belonging to the Janus kinase (JAK) family. Specifically, the mammalian JAK…

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Posted in: Acanthosis, Colitis, Systemic Lupus Erythematosus Filed under: CYP2C19, Tyk2

BMS-986251 is an Orally Active and Selective RORγt Inverse Agonist

2020-07-07 Edward Jenner

Retinoic acid-related orphan receptor γt (RORγt) is a nuclear hormone receptor (NHR) and belongs to the RORγ family. It exists…

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Posted in: Autoimmune Disorders, Inflammation, Skin Inflammation Filed under: Acanthosis, IL-17, RORγ

CCG-203971 is a Second-Generation RhoA/MRTF-A Inhibitor with Antifibrotic Effect

2020-03-21 Edward Jenner

Metastasis is the major driver in cancer-related deaths. Metastases involve dysregulation of numerous cellular processes. Importantly, blockade of RhoC prevents…

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Posted in: Fibrosis, Systemic Scleroderma Filed under: MRTF, RhoA, SRF

AS2863619, a Foxp3 Inducer, is an Orally Active CDK8/19 Inhibitor

2019-11-28 Edward Jenner

AS2863619 is a potent, orally active cyclin-dependent kinase 8 (CDK8) and CDK19 inhibitor with IC50s of  0.61 nM and 4.28 nM, respectively. Firstly, in vitro,…

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Posted in: Allergy, Skin Inflammation Filed under: CDK, GSK3

Remibrutinib is an Orally Active BTK Inhibitor for the Chronic Urticaria Treatment

2019-11-09 Edward Jenner

Chronic urticaria is a heterogeneous, persistent, and severely debilitating disease. Bruton’s tyrosine kinase (BTK) is a non-receptor kinase that plays…

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Posted in: Allergy, Chronic Urticaria, Skin Inflammation Filed under: Btk

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