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Immune System Research

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TC-2153 is STEP Inhibitor with Psychotropic Activity and Low Acute Toxicity

Edward Jenner 2023-04-21

Striatal-enriched protein tyrosine phosphatase (STEP) is a CNS-rich protein associated with a variety of neurological and neuropsychiatric disorders. Firstly, it is expressed exclusively in the central nervous system. Then, it…

Alzheimer Epilepsy Inflammation Ischemia Multiple Sclerosis Neurological Disease

Fuzapladib (IS-741) is A Potent Phospholipase A2 Inhibitor

Edward Jenner 2023-02-16

Phospholipase is a member of a very complex group of enzymes that break down phospholipids into fatty acids and other compounds. Phospholipase is defined by the enzymatic reaction they catalyze.…

Alzheimer Inflammation Neurological Disease Parkinson’s

SB26019, An Anti-Neuroinflammatory Agent, Induces Monomeric α-tubulin Formation

Edward Jenner 2023-02-08

Nuclear factor kappa B (NF-κB) family transcription factors are the master regulators. NF-κB is indispensable for a wide variety of biological processes including inflammation and the immune system. NF-kB functions…

Alzheimer Parkinson’s

DN-1289 is an Orally Active and Selective Inhibitor of DLK and LZK

Edward Jenner 2023-01-20

Double leucine zipper kinase (DLK, MAP3K12) and leucine zipper Carrying kinase (LZK, MAP3K13) are two homologous mitogen-activated protein kinases. They are regulators of neuronal apoptosis and axon degradation. And also…

Alzheimer Antibodydrug Neurological Disease

Semorinemab (RG 6100) is an Anti-Tau Humanized IgG4 Monoclonal Antibody

Edward Jenner 2023-01-09

Tau (Tubulin-associated unit) is a microtubule-associated protein (MAP) that is primarily present in axons. Besides, Tau is a multi-functional protein. Particularly, It takes part in the cross-linking and regulation of…

Alzheimer Inflammation Neuroimmunology

VQW-765 (AQW-051) is a Selective and Orally Active α7-nAChR Agonist

Edward Jenner 2022-12-28

nAChRs (nicotinic acetylcholine receptors) are neuron receptor proteins that signal for muscular contraction upon a chemical stimulus. In mammals, analysis of cDNA proved existence of 17 homologues of nAChR's subunits…

Alzheimer Inflammation Neurological Disease

SZM679 is an Orally Active and Selective RIPK1 Inhibitor, Can be Used to Research Alzheimer\’s Disease

Edward Jenner 2022-12-16

RIPK1 (Receptor-interacting serine/threonine-protein kinase 1), a 76-kDa protein, is an essential mediator of cell death and inflammation. This protein has a N-terminal kinase domain, a C-terminal death domain, and an…

Alzheimer Neurological Disease Parkinson’s

Virodhamine, an Endocannabinoid, Regulates Neurotransmission

Edward Jenner 2022-12-02

The endogenous cannabinoid system consists of endogenous cannabinoids, cannabinoid receptors, and enzymes that synthesize and degrade endogenous cannabinoids. Specifically, many effects of cannabinoids and endogenous cannabinoids are mediated by two…

Alzheimer Neuroimmunology Neurological Disease Parkinson’s

AMS-17 is a Potent NLRP3 Inhibitor, Inhibiting Microglia Activation

Edward Jenner 2022-07-07

Microglia is a kind of resident immune cell in the central nervous system (CNS) parenchyma. microglia remain in a quiescent state Under normal physiological conditions. Besides, Brain injury and some…

Alzheimer

Elenbecestat (E2609) is an Orally Active and CNS-penetrant BACE-1 Inhibitor

Edward Jenner 2022-05-26

AAlzheimer's disease (AD)  is a neurodegenerative disease, characterized by progressive memory loss. In AD patients' brain, the Aβ-containing plaques and tau-containing neurofibrillary tangles exhibit significant accumulation. Aβ is primarily generated…

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You Missed

Cancer Chronic Urticaria Inflammatory Uncategorized

Remibrutinib is an Orally Active BTK Inhibitor for Chronic Urticaria Research

Infection

Taurolidine is a Broad-spectrum Antimicrobial for Central Venous Catheter-Related Infections Research

Endocrinology Parkinson’s

Cabergoline is a D2-like Receptor Agonist for High Prolactin Levels Related Diseases

Inflammation

Ondansetron is a 5-HT3 Receptor Antagonist for Anti-inflammation Research

Immune System Research

Up to date immunology information

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