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Category: Arthritis

UCB-9260 Inhibits TNF Signalling by Stabilising an Asymmetric form of the Trimer

2021-02-10 Edward Jenner

Tumor necrosis factor (TNF) is a cytokine belonging to a family of trimeric proteins. This factor acts as a key…

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Posted in: Arthritis, Collagen-Induced Arthritis Filed under: CAIA, TNF

GSK620 is a Potent and Orally Active pan-BET-BD2 Inhibitor

2021-01-08 Edward Jenner

The therapeutic potential of extra terminal domain inhibitor (iBET) has increasing studies both in oncology and immunoinflammatory. Moreover, iBETs are…

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Posted in: Arthritis, Hepatitis, Inflammation, Psoriasis Filed under: Anti-Inflammatory, BET BD2, BRD4, Psoriasis

HS271 is a Highly Potent, Orally Active and Selective IRAK4 Inhibitor

2020-12-24 Edward Jenner

IRAK-4 (interleukin-1 receptor-associated kinase 4) is a protein kinase involved in signal transduction of innate immune response from toll-like receptors.…

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Posted in: Arthritis, Collagen-Induced Arthritis Filed under: Antiinflammatory, IRAK4, TNFα

SP-100030 is a Potent NF-κB and Activator Protein-1 (AP-1) Inhibitor

2020-10-01 Edward Jenner

Nuclear factor-κB (NF-κB) represents a family of inducible transcription factors. The transcription factor NF-κB regulates multiple aspects of innate and…

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Posted in: Arthritis, Collagen-Induced Arthritis, Inflammation Filed under: AP-1, Interleukin, Jurkat, NF-κB, TNF-α

RVX-297 is an Orally Bioavailable and Selective BET BD2 Inhibitor

2020-07-22 Edward Jenner

Proinflammatory stimuli induce rapid transcriptional responses. They are essential for host defense from infection. An inflammatory response involves a variety…

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Posted in: Arthritis, Autoimmune Disorders, Collagen-Induced Arthritis, Inflammation Filed under: BET BD2, Bromodomain, IL-6

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