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Immune System Research
Up to date immunology information.

Category: Neurological Disease

DN-1289 is an Orally Active and Selective Inhibitor of DLK and LZK

2023-01-20 Edward Jenner

Double leucine zipper kinase (DLK, MAP3K12) and leucine zipper Carrying kinase (LZK, MAP3K13) are two homologous mitogen-activated protein kinases. They…

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Posted in: Alzheimer, Parkinson’s Filed under: Alzheimer´s Disease, amyotrophic lateral sclerosis, DLK, DN-1289, JNK, LZK, Parkinson's disease

Semorinemab (RG 6100) is an Anti-Tau Humanized IgG4 Monoclonal Antibody

2023-01-09 Edward Jenner

Tau (Tubulin-associated unit) is a microtubule-associated protein (MAP) that is primarily present in axons. Besides, Tau is a multi-functional protein.…

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Posted in: Alzheimer, Antibodydrug, Neurological Disease Filed under: Alzheimer´s Disease, Anti-Tau, Monoclonal Antibody

VQW-765 (AQW-051) is a Selective and Orally Active α7-nAChR Agonist

2022-12-28 Edward Jenner

nAChRs (nicotinic acetylcholine receptors) are neuron receptor proteins that signal for muscular contraction upon a chemical stimulus. In mammals, analysis…

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Posted in: Alzheimer, Inflammation, Neuroimmunology Filed under: Anxiolytic, Cognitive disorders, learning/memory performance

ZZL-7 is a Fast-Onset Antidepressant Agent

2022-12-23 Edward Jenner

Serotonin Transporters (SERTs) are integral membrane proteins that transport serotonin from synaptic spaces into presynaptic neurons. SERTs function by reuptake…

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Posted in: Neurological Disease Filed under: Antidepressant, Major Depressive Disorder, nNOS, SERT

Ph-HTBA is a Brain-Penetrating CaMKIIα Modulator and Used for The Research of Neurodegenerative Disorders

2022-12-22 Edward Jenner

CaMKII (Ca2+/calmodulin-dependent protein kinase II) is an oligomeric protein kinase assembled by 12−14 monomers in a double-layered ring. Structurally, each…

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Posted in: Cognitive Disorders, Neurological Disease Filed under: Brain-penetrant, CaMKIIα, Neuroprotective

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