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Diabetes Diabetes Type 2 Diabetes Mellitus

AZD1092 is an Orally Active GK Activator for the Research of Type 2 Diabetes

Edward Jenner 2023-07-24

Glucokinase is a hexokinase isozyme that facilitates phosphorylation of glucose to glucose-6-phosphate. This is the rate-limiting step in glucose metabolism. Glucokinase occurs in cells in the liver and pancreas of…

Diabetes Diabetes Neurological Disease

BT44 is an RET Activator for Neurodegenerative Disorders and Diabetes Mellitus Research

Edward Jenner 2023-06-07

The glial cell line-derived neurotrophic factor (GDNF) family ligands (GFLs) alleviate symptoms of experimental neuropathy, protect and stimulate the regeneration of sensory neurons in animal models of neuropathic pain, and…

Diabetes Diabetes

SB-435495 is an Orally Active Lp-PLA2 Inhibitor for Diabetes Research

Edward Jenner 2023-06-01

Lp-PLA2 (Lipoprotein-associated phospholipase A2) is a calcium-independent serine lipase of 50-kDa that hydrolyzes the acetyl group at the sn-2 position of the platelet-activating factor. Importantly, Lp-PLA2 circulates in plasma bound…

Diabetes Diabetes

Empagliflozin (BI 107730) is a Selective SGLT-2 Inhibitor for Type 2 Diabetes Research

Edward Jenner 2023-03-01

Diabetes has a major impact on the global human population. Generally, blood glucose control is the major method of diabetes treatment. Previous studies indicated that targeting sodium glucose co-transporter-2 (SGLT-2)…

Diabetes Diabetic Complication

Midaglizole is a Potent α2-Adrenoceptor Antagonist with a Hypoglycemic Activity

Edward Jenner 2023-02-13

α2-adrenoceptor is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. Besides, the α2-adrenoceptor not only inhibits the release of their neurotransmitters (autoreceptors) but can also regulate the…

Recent Posts

  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
  • Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research
  • Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research
  • Doravirine is a HIV-1 Inhibitor for Infection Research

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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