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Immune System Research
Up to date immunology information.

Category: Innate Immune

GDC-2394 is an Orally Active and Selective NLRP3 Inhibitor

2022-11-24 Edward Jenner

Nucleotide oligomerization domain (NOD)-like receptors (NLRs) are critical cytoplasmic pattern-recognition receptors (PRRs) that play an important role in the host’s…

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Posted in: Immunology, Innate Immune Filed under: Anti-inflammatory Effect, IL-18, IL-1β, NLRP3

TAK-676 is a STING Agonist and Triggers the STING Signaling Pathway Activation

2022-09-03 Edward Jenner

Stimulator of interferon genes (STING), an integral ER-membrane protein, is a protein that in humans is encoded by the STING1…

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Posted in: Cancer Immunotherapy, Immunotherapy, Innate Immune Filed under: Antitumor activity, Interferon, STING

T16A(inh)-C01 is an Inhibitor of TMEM16A (ANO1)

2022-08-11 Edward Jenner

Calcium-activated chloride channels (CaCCs) are always expressed in epithelial and nonepithelial cells. They are involved in epithelial fluid secretion, sensory…

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Posted in: hypertension, Inflammation, Innate Immune Filed under: Asthma, CaCCs, hypertension, Pain, secretory diarrheas, T16Ainh-A01, TMEM16A, tracheomalacia

SEW2871 is a Highly Selective and Orally Active S1P1 Agonist

2019-11-07 Edward Jenner

G protein-coupled receptors (GPCRs) are also known as 7TM receptors due to their transmembrane domains. they constitute the largest superfamily…

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Posted in: Colitis, Fibrosis, Inflammation, Innate Immune Filed under: IL-10, Interleukin, S1P

C-178 is a Covalent Small-Molecule Inhibitor of STING

2019-09-26 Edward Jenner

In the previous blog, I have introduced C-176 as a strong and covalent mouse STING inhibitor. Today, I’d like to…

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Posted in: Autoimmune Disorders, Inflammation, Innate Immune Filed under: Interferon, STING

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