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Category: Rheumatoid Arthritis

LS-102 is a Selective Synoviolin (Syvn1) Inhibitor

2020-04-14 Edward Jenner

Rheumatoid arthritis (RA) is the most common chronic inflammatory joint disease, affecting many people in the industrialized world. Synoviolin (Syvn1)…

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Posted in: Arthritis, Rheumatoid Arthritis Filed under: Autoubiquitination, E3 Ligase, Synoviolin, Syvn1

J-113863 is a CCR1 Antagonist for Rheumatoid Arthritis Treatment

2020-02-12 Edward Jenner

The CC-type chemokine receptor 1 (CCR1) is a chemokine receptor of significant importance in human health. CCR1 is a protein…

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Posted in: Arthritis, Rheumatoid Arthritis Filed under: Anti-Inflammatory, CCR1, CCR3, Chemokines

Rofecoxib is a Specific and Orally Active COX-2 Inhibitor for Rheumatoid Arthritis Treatment

2019-12-25 Edward Jenner

Cyclooxygenase (COX) -2 is an inducible form of COX, and it involves in inflammation. In addition, Malignant mesothelioma (MM) is…

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Posted in: Rheumatoid Arthritis Filed under: Anti-Inflammatory, COX

Upadacitinib is an Orally Active and Selective JAK1 Inhibitor

2019-12-22 Edward Jenner

Biologic agents are highly effective therapies. It greatly improves the standard of care for patients with rheumatoid arthritis (RA). Even…

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Posted in: Arthritis, Autoimmune Disorders, Rheumatoid Arthritis Filed under: Anemia, JAK1

C25-140 is a Selective TRAF6-Ubc13 Inhibitor to Combate Autoimmunity

2019-09-28 Edward Jenner

The TRAF protein family comprises seven E3 ligase members, including TRAF6. Distinct receptor signaling pathways have different members, such as…

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Posted in: Autoimmune Disorders, Rheumatoid Arthritis Filed under: Autoimmunity, TRAF, Ubc13

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