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Category: Hepatitis

Grazoprevir is a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease

2021-12-21 Edward Jenner

Hepatitis C virus (HCV) is a member of the Flaviviridae family of viruses in the Hepacivirus genus. Meanwhile, HCV NS3-4A…

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Posted in: Hepatitis, Hepatitis C Virus Filed under: HCV, HCV NS3, Hepatitis

PF-05221304 is an Orally Active, Liver-Directed and Dual ACC1 (and ACC2) Inhibitor

2021-03-17 Edward Jenner

The character of nonalcoholic fatty liver disease (NAFLD) is the accumulation of fat (in excess of 5%) within the hepatocytes.…

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Posted in: Hepatitis Filed under: ACC1, ACC2, CDAHFD, NAFL, NASH

GSK620 is a Potent and Orally Active pan-BET-BD2 Inhibitor

2021-01-08 Edward Jenner

The therapeutic potential of extra terminal domain inhibitor (iBET) has increasing studies both in oncology and immunoinflammatory. Moreover, iBETs are…

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Posted in: Arthritis, Hepatitis, Inflammation, Psoriasis Filed under: Anti-Inflammatory, BET BD2, BRD4, Psoriasis

BA-53038B is a HBV Core Protein Allosteric Modulator (CpAM)

2019-07-01 Edward Jenner

In our previous blogs, we have introduced two HBV inhibitors. Today, I’d like to describe another small molecule compound BA-53038B…

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Posted in: Chronic Hepatitis B, Viral Immunology Filed under: Antiviral, HBV
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