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Immune System Research
Up to date immunology information.

Category: Complement System

Narsoplimab (OMS 721) is an IgG4 mAb That Binds MASP-2 and Blocks Lectin Pathway Activation

2023-01-23 Edward Jenner

MASP-2 (Mannan-binding lectin-associated serine protease-2) is a key serine protease in the lectin pathway of complement activation, resulting in excessive…

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Posted in: Antibodydrug, Complement System, SARS-CoV-2 Filed under: anti-MASP-2, HSCT, MASP-2, Monoclonal Antibody, SARS-CoV-2

Pegcetacoplan is a Pegylated Complement C3 Inhibitor Peptide

2022-11-19 Edward Jenner

Complement component 3 is a protein of the immune system that contains 13 structural domains. C3 plays an important role…

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Posted in: Autoimmune Encephalomyelitis, Complement System Filed under: C3b, complement C3, Haemolytic anaemia, Paroxysmal nocturnal hemoglobinuria

Zilucoplan (RA101495) is a Potent Complement Component 5 Inhibitor

2022-11-12 Edward Jenner

The complement system, composed of more than 30 serum and cell surface components, is collaborating in the recognition and elimination…

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Posted in: Complement System Filed under: C5, Complement Component 5, Immune-mediated Necrotising Myopathy, Myasthenia Gravis

PMX-53 is an Orally Active Complement C5a Receptor Antagonist

2020-06-09 Edward Jenner

C5a is an important inflammatory hypernociceptive mediator, acting by a mechanism independent of hypernociceptive cytokine release, but dependent on the…

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Posted in: Allergy, Complement System, Inflammation Filed under: Anti-Tumor, Antiatherosclerotic, C5a, CD88

MK-0429 is An Oral Integrin (αvβ3) Inhibitor

2019-04-11 Edward Jenner

Integrins are cell surface protein receptors with α and β subunits. They participate in multiple cellular functions such as adhesion…

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Posted in: Cancer Immunology, Complement System, Kidney Fibrosis Filed under: Integrin
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