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Category: Rheumatoid Arthritis

Tenidap, a Non-Steroidal Anti-Inflammatory Drug, is a Selective COX-1 Inhibitor

2022-03-17 Edward Jenner

Cyclooxygenase (COX) is a key step in the conversion of arachidonic acid to PGH2. Specifically, PGH2 is a direct substrate…

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Posted in: Inflammation, Rheumatoid Arthritis Filed under: Antirheumatic, COX-1, SLC26A3

PF06650833 is an Orally Active IRAK4 Inhibitor

2020-09-15 Edward Jenner

Interleukin-1 receptor-associated kinase 4 (IRAK4) is a key node in innate inflammatory signaling. It is also directly downstream of the…

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Posted in: Rheumatoid Arthritis Filed under: Anti-Inflammatory, IRAK4, Lupus, Lymphomas

PF-9184 is a Highly Selective of Human Microsomal PGES-1 Inhibitor

2020-08-04 Edward Jenner

mPGES-1 is the terminal enzyme one-step downstream of COX2. It also is the unstable peroxide intermediate from arachidonate catabolism. mPGES-1…

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Posted in: Rheumatoid Arthritis Filed under: IL-1β, PGE, PGES, RASF, TXB2

MS417 is a BET-Specific BRD4 Inhibitor

2020-01-17 Edward Jenner

NF-κB-mediated inflammation is a major pathology in kidney diseases, such as non-kidney inflammatory diseases, and rheumatoid arthritis. HIV infection in…

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Posted in: HIV, Inflammation, Rheumatoid Arthritis, Viral Immunology Filed under: BRD4, HIV, HIVAN, NF-κB

E6130 is an Orally Active and Highly Selective CX3CR1 Modulator

2019-09-07 Edward Jenner

Infiltration of leukocytes from the peripheral circulation into tissues such as the gut mucosa is an important aspect of immune…

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Posted in: Colitis, Rheumatoid Arthritis Filed under: Anti-Inflammatory, CX3CR

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