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Arthritis Rheumatoid Arthritis

TAK-603 is a Potent and Orally Active Antirheumatic Agent for Adjuvant Arthritis Research

Edward Jenner 2023-06-21

Anti-arthritis drugs are used to relieve or prevent arthritis symptoms (such as joint pain and Joint stiffness). Specifically, the impact of rheumatism on fertility and reproduction may be significant. Individuals…

Inflammatory Rheumatoid Arthritis Skin Inflammation

GLPG2534 is an Orally Active IRAK4 Inhibitor for Inflammatory Skin Diseases Research

Edward Jenner 2023-06-02

Kinases typically integrate signaling events down-stream of multiple cytokine receptors. Hence, kinase inhibitors distinguish themselves from cytokine-targeted biologicals by their capacity to modulate multiple signaling pathways simultaneously. IL-1 receptor (IL-1R)–associated…

Immune Rheumatoid Arthritis

PPI-2458 is an Orally Active and Irreversible MetAP-2 Inhibitor for Tumor Research

Edward Jenner 2023-03-02

MetAP-2, a cytoplasmic metalase, catalyzes the hydrolysis and removal of N-terminal methionine residues from newborn proteins. The enzymatic activity of MetAP-2 is a prerequisite for biological processes such as activity,…

Inflammation Rheumatoid Arthritis

Salubrinal is a cell-permeable and selective inhibitor of eIF2α dephosphorylation

Edward Jenner 2023-01-04

eIF2 (eukaryotic initiation factor 2), an eukaryotic initiation factor, is an essential factor for protein synthesis. eIF2 mediates the binding of tRNAiMet to the ribosome in a GTP-dependent manner. And…

Rheumatoid Arthritis

Fletikumab (NNC0109-0012) is a Monoclonal Antibody Targeting IL-20

Edward Jenner 2022-10-27

IL-20 (Interleukin-20) is a member of IL-10 family, which includes IL-10, IL-19, IL-22, IL-24, IL-26, IL-28, and IL-29. Besides, IL-20 is mainly produced by myeloid cells such as monocytes, granulocytes,…

Inflammation Rheumatoid Arthritis

Tenidap, a Non-Steroidal Anti-Inflammatory Drug, is a Selective COX-1 Inhibitor

Edward Jenner 2022-03-17

Cyclooxygenase (COX) is a key step in the conversion of arachidonic acid to PGH2. Specifically, PGH2 is a direct substrate for a series of cell-specific prostaglandin and thromboxane syntheses. Besides,…

Rheumatoid Arthritis

PF06650833 is an Orally Active IRAK4 Inhibitor

Edward Jenner 2020-09-15

Interleukin-1 receptor-associated kinase 4 (IRAK4) is a key node in innate inflammatory signaling. It is also directly downstream of the Toll-like receptors (TLRs) and interleukin-1 (IL-1) family of receptors. Besides,…

Rheumatoid Arthritis

PF-9184 is a Highly Selective of Human Microsomal PGES-1 Inhibitor

Edward Jenner 2020-08-04

mPGES-1 is the terminal enzyme one-step downstream of COX2. It also is the unstable peroxide intermediate from arachidonate catabolism. mPGES-1 can be induced by various inflammatory stimuli in normal cells,…

HIV Inflammation Rheumatoid Arthritis Viral Immunology

MS417 is a BET-Specific BRD4 Inhibitor

Edward Jenner 2020-01-17

NF-κB-mediated inflammation is a major pathology in kidney diseases, such as non-kidney inflammatory diseases, and rheumatoid arthritis. HIV infection in the kidney induces NF-κB activation, leading to the production of…

Colitis Rheumatoid Arthritis

E6130 is an Orally Active and Highly Selective CX3CR1 Modulator

Edward Jenner 2019-09-07

Infiltration of leukocytes from the peripheral circulation into tissues such as the gut mucosa is an important aspect of immune surveillance. They interact with cytokine or other proinflammatory stimuli-activated endothelial…

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

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