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Immune System Research
Up to date immunology information.

Category: Cognitive Disorders

Ph-HTBA is a Brain-Penetrating CaMKIIα Modulator and Used for The Research of Neurodegenerative Disorders

2022-12-22 Edward Jenner

CaMKII (Ca2+/calmodulin-dependent protein kinase II) is an oligomeric protein kinase assembled by 12−14 monomers in a double-layered ring. Structurally, each…

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Posted in: Cognitive Disorders, Neurological Disease Filed under: Brain-penetrant, CaMKIIα, Neuroprotective

SSR504734 is an Orally Active, Selective and Reversible GlyT1 Inhibitor

2022-09-22 Edward Jenner

Glycine transporters (GlyTs) are the Na+/Cl–-dependent plasmalemmal neurotransmitter transporters. GlyTs comprise GlyT1 and GlyT2. They serve to terminate the signaling…

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Posted in: Analgesia, Cognitive Disorders, Epilepsy, Neurological Disease, Schizophrenia Filed under: Anti-anxiety, Anti-depression, Anti-schizophrenia

ATC0175 is a Potent, Selective and Orally Active MCH1R Antagonist.

2022-07-28 Edward Jenner

MCH1R (melanin-concentrating hormone 1 receptor) is one of the melanin-concentrating hormone receptors found in all mammals. What\’s more, The protein…

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Posted in: Cognitive Disorders, Neurological Disease Filed under: Anxiety, Depression, MCH1R

Blonanserin is a Potent and Orally Active 5-HT2A and Dopamine D2 Receptor Antagonist

2022-07-26 Edward Jenner

5-HT receptors (Serotonin receptors) are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs). They mediate both…

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Posted in: Cognitive Disorders, Neurological Disease, Uncategorized Filed under: Antidepression, Antipsychotic agent

Mirogabalin is a Selective and Orally Active Ligand for the α2δ Subunit of Voltage-Gated Calcium Channels

2022-05-14 Edward Jenner

Voltage-gated calcium channels (VGCC) are a group of voltage-gated ion channels in the membrane of excitable cells. Specifically, they have…

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Posted in: Cognitive Disorders, Neurological Disease Filed under: calcium channel, VGCC

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