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FDA Approves Lotilaner for the Research of Demodex Blepharitis

Edward Jenner 2023-08-15

GABA (γ-aminobutyric acid-gated) is the chief inhibitory neurotransmitter in the developmentally mature mammalian central nervous system. Besides, Its principal role is reducing neuronal excitability throughout the nervous system. GABACl (γ-aminobutyric…

Malaria Parasite

DSM705 is a Plasmodium DHODH Inhibitor

Edward Jenner 2021-06-30

Malaria is one of the most widespread and ancient infectious diseases of humanity. In particular, Dihydroorotate dehydrogenase (DHODH) acts as a target for the development of new antimalarials. In addition,…

Infection Parasite

Melarsomine, an Adulticide, is Used in the Canine Heartworm Disease Study

Edward Jenner 2021-04-15

Dirofilaria repens is a filarial parasite of canids transmitting by mosquitoes. Besides, adult worms mainly exist in the subcutaneous tissue of dogs. And it deposits microfilariae that circulate in the…

Malaria Parasite

SJ000025081, a Dihydropyridine, Acts as a Potent Antimalarial Agent

Edward Jenner 2020-10-17

Malaria is a mosquito-borne infectious disease that affects humans and other animals. Specifically, malaria caused Symptoms usually including fever, fatigue, vomiting and headache. Besides, malaria is due to the single-celled…

Malaria Parasite

AN3661, an Antimalarial Agent, is a PfCPSF3 Inhibitor

Edward Jenner 2020-06-11

Cleavage and polyadenylation specificity factor (CPSF) is relevant to the cleavage of the 3' signaling region from a newly synthesized pre-messenger RNA (pre-mRNA) molecule. Specifically, it is in the process…

Parasite

KDU731, a PI4K inhibitor, Blocks Cryptosporidium Infection

Edward Jenner 2019-10-09

The apicomplexan parasite Cryptosporidium is one of the leading causes of infectious diarrhea in children. Cryptosporidiosis is also a well-recognized opportunistic infection in adult AIDS and transplant patients. The Cryptosporidium…

Malaria Parasite

TCMDC-135051, a Highly Selective PfCLK3 Inhibitor, Has Potential to Treat Malaria

Edward Jenner 2019-09-20

PfCLK3 is a protein kinase essential for maintaining the asexual blood stage of both P. falciparum and P. berghei.  In mammalian cells, the CLK protein kinase family and the closely related SRPK family…

Cancer Immunology Immune Checkpoint Parasite

RRx-001 is a Dual Checkpoint Inhibitor by Downregulating CD47 and SIRP-α

Edward Jenner 2019-09-08

As previously introduced, we all have known that RRx-001, a hypoxia-selective epigenetic agent and a radio- and chem-sensitizer. Additionally, it triggers apoptosis and overcomes drug resistance in myeloma. RRx-001 exhibits…

Parasite

BKI-1369 is an Effective Bumped Kinase Inhibitor with Anti-Cryptosporidiosis Effect

Edward Jenner 2019-08-25

Nowadays, cryptosporidiosis is no stranger to us. We have mentioned such disease in our previous blogs. It is a main cause of diarrhea in children under 2 years old especially…

Parasite

AN7973 Blocks Intracellular Parasite Development to Treat Cryptosporidiosis

Edward Jenner 2019-08-17

Cryptosporidiosis is a kind of parasitic diseases, caused by Cryptosporidium. The parasite commonly exists in HIV-positive patients. It is harmful to the distal small intestine and affects the respiratory tract…

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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