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Autoimmune diseases Inflammatory

SZM-1209 is an Orally Active RIPK1 Inhibitor with Anti-SIRS and Anti-ALI Effects

Edward Jenner 2023-05-11

Receptor-interacting protein (RIP) kinases are a group of threonine/serine protein kinases. There are seven members of the RIPK family, RIPK1-7. RIP kinases are cellular signaling molecules that are critical for…

Autoimmune diseases Inflammatory Uncategorized

SRTCX1003 is an Orally Active SIRT1 Activator for Inflammatory Research

Edward Jenner 2023-04-19

Sirtuin (Sir2 proteins) is a class of proteins. And it possesses either mono-ADP-ribosyltransferase, or deacylase activity, including deacetylase, desuccinylase, demalonylase, demyristoylase and depalmitoylase activity. Sirtuins regulate important biological pathways in…

Autoimmune diseases

Deucravacitinib is an Orally Active TYK2 Allosteric Inhibitor for Autoimmune Diseases Research

Edward Jenner 2023-04-11

Tyrosine kinase 2 (TYK2) is a member of the JAK kinase family. Besides, it regulates signal transduction downstream of the IL-23/IL-12 pathway and the type I interferon family receptor, pairing…

Autoimmune diseases Graves' hyperthyroidism Inflammation

Iscalimab (CFZ-533) is an IGg1 mAb Targeting CD40 for Inflammation Research

Edward Jenner 2023-03-13

CD40 is a transmembrane glycoprotein. CD40 can express on B cells and antigen presenting cells (APCs) such as monocytes, macrophages, and dendritic cells (DC). It also expresses on platelets. Furthermore, …

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  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

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