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Infection Malaria Parasite

UCB7362 is an Orally Active Antimalarial Plasmepsin X Inhibitor

Edward Jenner 2022-11-15

Malaria is a parasitic disease caused by Plasmodium species, which are spread by mosquitoes. The parasites enter the bloodstream through the mosquito's saliva, then live in the liver to develop and…

Fungal Infection Parasite

Oleandomycin is a Macrolide Antibiotic

Edward Jenner 2022-04-14

Antibiotics are antibacterial substances that are active against bacteria. Antibiotics have an effect on treating and preventing such infections. Meanwhile, they can kill or inhibit the growth of bacteria. A…

Infection Inflammation Parasite

Diminazene aceturate is an Anti-trypanosome Agent for Animals

Edward Jenner 2022-04-01

Trypanosomiasis or trypanosomosis is the name of several diseases in vertebrates caused by parasitic protozoan trypanosomes of the genus Trypanosoma. A number of these diseases occur in animals. Trypanosomiasis in…

Infection Inflammation Parasite

PK 11195 is a Ligand of Translocator Protein (TSPO) for Leishmania Chemotherapy

Edward Jenner 2022-02-12

PK 11195, a ligand of this protein, acts as an anti-leishmanial agent. At the same time, PK 11195 exhibits IC<sub>50</sub> values of 14.2 μM for L. amazonensis, 8.2 μM for…

Infection Parasite

LXE408 is an Orally Active Proteasome Inhibitor with Anti-leishmaniasis Activity

Edward Jenner 2020-08-22

Proteasomes are protein complexes that degrade unwanted or damaged proteins by proteolysis, which can destroy peptide bonds. Specifically, proteasomes are part of the main mechanism by which cells regulate the…

Infection Parasite

NPD1335 is a Trypanosoma Brucei Phosphodiesterase B1 Inhibitor

Edward Jenner 2019-08-22

Trypanosoma brucei (T.b.) rhodesiense and T.b. gambiense are endemic in sub-Saharan Africa. They are typical two causative agents of human African trypanosomiasis (HAT). The drugs for HAT treatment currently on…

Recent Posts

  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
  • Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research
  • Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research
  • Doravirine is a HIV-1 Inhibitor for Infection Research

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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