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Immune System Research
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Category: Malaria

WM382 is an Orally Active Plasmepsin IX/X Inhibitor with Antimalarial Activity

2022-12-01 Edward Jenner

Malaria is a parasitic disease caused by Plasmodium species, which are spread by mosquitoes. Erythrocytes are the replicating factories for malaria…

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Posted in: Infection, Malaria Filed under: Antimalarial, aspartic protease, Malaria, Parasite, Plasmepsin, WM382

UCB7362 is an Orally Active Antimalarial Plasmepsin X Inhibitor

2022-11-15 Edward Jenner

Malaria is a parasitic disease caused by Plasmodium species, which are spread by mosquitoes. The parasites enter the bloodstream through the…

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Posted in: Infection, Malaria, Parasite Filed under: Malaria, Plasmepsin, Plm X

Manzamine A, an Orally Active β-carboline Alkaloid, Inhibits GSK-3β and CDK-5

2021-07-29 Edward Jenner

Glycogen synthase kinase-3 (GSK-3) is a serine-threonine kinase ubiquitously expressed and involved in the regulation of many cell functions. GSK-3…

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Posted in: Cancer Immunology, Inflammation, Malaria Filed under: Antimalarial, ATPase, Autophagy, CDK-5, GSK-3β, HSV-1

DSM705 is a Plasmodium DHODH Inhibitor

2021-06-30 Edward Jenner

Malaria is one of the most widespread and ancient infectious diseases of humanity. In particular, Dihydroorotate dehydrogenase (DHODH) acts as…

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Posted in: Malaria, Parasite Filed under: Antimalarial, DHODH, Parasite

FNDR-20123 is an Orally Active and a First-in-Class Anti-Malarial HDAC Inhibitor

2021-03-20 Edward Jenner

Malaria remains one of the most severe and life-threatening infectious diseases. Among the various Plasmodium spp., Plasmodium falciparum is the most…

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Posted in: Malaria Filed under: Antimalarial, HDAC

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