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ER-27319 is a Syk Inhibitor for Inflammation Diseases Research

Edward Jenner 2023-09-14

Inflammation involving the innate and adaptive immune systems is a normal response to infection. However, when allowed to continue unchecked, inflammation may result in autoimmune or autoinflammatory disorders, neurodegenerative disease,…

Cancer Immunology Immunology

Diprovocim is a Potent TLR1/TLR2 Agonist

Edward Jenner 2022-12-30

Toll-like receptors (TLRs) play a crucial role in the innate immune system by recognizing pathogen-related molecular patterns from various microorganisms. Specifically, TLRs signal by recruiting specific adaptor molecules, leading to…

Immunology

RI-962 is a Selective RIPK1 Inhibitor for Inflammatory Diseases Research

Edward Jenner 2022-12-17

RIPK1 (receptor-interacting protein kinase 1) is a serine/threonine protein kinase. It also is a key regulator of programmed cell necrosis (necroptosis). RIPK1 is closely related to the occurrence and development…

Immunology Innate Immune

GDC-2394 is an Orally Active and Selective NLRP3 Inhibitor

Edward Jenner 2022-11-24

Nucleotide oligomerization domain (NOD)-like receptors (NLRs) are critical cytoplasmic pattern-recognition receptors (PRRs) that play an important role in the host's innate immune response and immunity homeostasis. Additionally, Members of the…

Immunology

SLF1081851 is a Potent Spns2 Inhibitor

Edward Jenner 2022-09-24

Spns2 (Sphingolipid Transporter 2) is a non-ATP dependent S1P (sphingosine-1-phosphate) transporter, that transports S1P from endothelial and lymph-endothelial cells, and regulates S1P concentration in plasma and lymph. Particularly, Sphingosine 1-phosphate…

Endocrinology Immunology

CHF-6366 is a M3 Muscarinic Antagonist and β2-adrenergic Receptors Agonist

Edward Jenner 2022-09-15

Muscarinic receptor, also known as muscarinic cholinergic/acetylcholine receptor (mAChR), belongs to the G protein-coupled receptor (GPCR) family and is found in many parts of the body, such as brain and…

Immunology Immunotherapy Inflammation

Perindoprilat (S 9780) is an ACE inhibitor for Hypertension Research

Edward Jenner 2022-08-07

Perindoprilat (S 9780) is an angiotensin-converting enzyme (ACE) inhibitor with an IC50 value ranging from 1.5 nM. Besides, Perindoprilat shows an affinity for bradykinin and angiotensin I with specific binding rates of 47%…

Allergy Immunology Inflammation

Tecastemizole, A Major Metabolite of Astemizole, is a Potent and Selective H1 receptor Antagonist

Edward Jenner 2022-07-02

Histamine Receptors are a class of G protein-coupled receptors with histamine as their endogenous ligand. There are four types histamine receptors, H1R, H2R, H3R, and H4R. Histamine receptors play a…

Immunology

MRS 1754 is a Selective Antagonist Radioligand for A2B Adenosine Receptor

Edward Jenner 2022-04-26

Adenosine receptors (ARs) comprise a group of G protein-coupled receptors (GPCR) which mediate the physiological actions of adenosine. To date, there are four types of adenosine receptors in humans: A1,…

Immunology Inflammation Psoriasis Skin Inflammation

Secukinumab (AIN457) is a Human Monoclonal Antibody Targeted against IL-17A

Edward Jenner 2021-06-26

Interleukin-17 family (IL-17 family) is a pro-inflammatory cystine node cytokine family. After binding to the receptor, IL-17 can activate several signal cascades, leading to the induction of chemokines. As chemokines,…

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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