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Atopic Dermatitis Psoriasis

Tapinarof is an AhR Agonist for Skin Inflammation Research

Edward Jenner 2023-07-21

Aryl Hydrocarbon Receptor (AhR or AHR) is a cytoplasmic receptor and transcription factor that belongs to the family of basic helix-loop-helix transcription factors. The AhR is activated or inhibited by…

Inflammation Skin Inflammation

Tapinarof is a Natural Aryl Hydrocarbon Receptor (AhR) Agonist

Edward Jenner 2021-12-07

Tapinarof (GSK2894512) is a naturally-derived small molecule produced by bacterial symbionts of entomopathogenic nematodes. Especially, Tapinarof displays significant efficacy in psoriasis and atopic dermatitis (AD) modls. Psoriasis vulgaris is a…

Inflammation

VAF347 is a Highly Affinity Aryl Hydrocarbon Receptor (AhR) Agonist

Edward Jenner 2020-10-20

Aryl hydrocarbon receptor (AhR) are transcription factors that regulate gene expression. Specifically, AHR proteins contain several domains that are critical for their function. They are members of the basic helix…

Arthritis Rheumatoid Arthritis

CH-223191 Inhibits Smoking-Induced Aggravation of Experimental Arthritis via Aryl Hydrocarbon Receptor

Edward Jenner 2019-06-30

CH-223191 inhibits smoking-induced aggravation of experimental arthritis via aryl hydrocarbon receptor (AHR). Firstly, as we all know, smoking has become a major risk factor of people’s health. It involves in…

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You Missed

Cancer Chronic Urticaria Inflammatory Uncategorized

Remibrutinib is an Orally Active BTK Inhibitor for Chronic Urticaria Research

Infection

Taurolidine is a Broad-spectrum Antimicrobial for Central Venous Catheter-Related Infections Research

Endocrinology Parkinson’s

Cabergoline is a D2-like Receptor Agonist for High Prolactin Levels Related Diseases

Inflammation

Ondansetron is a 5-HT3 Receptor Antagonist for Anti-inflammation Research

Immune System Research

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