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Tag: Antimalarial

SJ000025081, a Dihydropyridine, Acts as a Potent Antimalarial Agent

2020-10-17 Edward Jenner

Malaria is a mosquito-borne infectious disease that affects humans and other animals. Specifically, malaria caused Symptoms usually including fever, fatigue,…

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Posted in: Malaria, Parasite Filed under: Antimalarial

AN3661, an Antimalarial Agent, is a PfCPSF3 Inhibitor

2020-06-11 Edward Jenner

Cleavage and polyadenylation specificity factor (CPSF) is relevant to the cleavage of the 3′ signaling region from a newly synthesized…

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Posted in: Malaria, Parasite Filed under: Antimalarial, CPSF3, PfCPSF3

TCMDC-135051, a Highly Selective PfCLK3 Inhibitor, Has Potential to Treat Malaria

2019-09-20 Edward Jenner

PfCLK3 is a protein kinase essential for maintaining the asexual blood stage of both P. falciparum and P. berghei.  In mammalian cells, the…

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Posted in: Malaria, Parasite Filed under: Antimalarial, CLK, Multidrug Resistance

RRx-001 is a Dual Checkpoint Inhibitor by Downregulating CD47 and SIRP-α

2019-09-08 Edward Jenner

As previously introduced, we all have known that RRx-001, a hypoxia-selective epigenetic agent and a radio- and chem-sensitizer. Additionally, it…

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Posted in: Cancer Immunology, Immune Checkpoint, Parasite Filed under: Antimalarial, CD47, SIRP-α

CWHM-1552 is an Orally Acitive Antimalarial Compound

2019-07-25 Edward Jenner

Malaria has been a military problem throughout history capable of causing epidemics that stop military operations. Particularly, malaria has had…

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Posted in: Malaria, Updated Filed under: Antimalarial, Infection

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