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Tag: EGFR

Toceranib (SU11654) is an Orally Active RTK Inhibitor

2022-06-23 Edward Jenner

Receptor tyrosine kinases (RTKs) are the high-affinity cell surface receptors for many polypeptide growth factors, cytokines, and hormones. In addition,…

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Posted in: Cancer Immunology Filed under: EGFR, Flt-3, KIT, Pdgfr, RTK, VEGFR

TAS6417 is a pan-Mutation Selective EGFR Inhibitor

2021-01-20 Edward Jenner

Despite dramatic response to first and second-generation EGFR TKIs, resistance emerges over time. The EGFR-T790M mutation accounts for more than…

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Posted in: Cancer Immunotherapy Filed under: EGFR, NSCLC, TKI

Neratinib is an Orally Available, Irreversible Tyrosine Kinase Inhibitor

2021-01-19 Edward Jenner

Neratinib is an irreversible tyrosine kinase inhibitor with IC50s of 59 nM and 92 nM for HER2 and EGFR, respectively.…

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Posted in: Cancer Immunotherapy Filed under: Breast Cancer, EGFR, HER

AG-1478 is a Selective EGFR Tyrosine Kinase Inhibitor

2021-01-16 Edward Jenner

Epidermal growth factor receptor (EGFR) is a transmembrane protein and a member of the ErbB receptor family. Specifically, EGFR is…

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Posted in: Cancer Immunotherapy, EMCV, HCV, Viral Immunology Filed under: A549, DU145, EGFR, EMCV, HCV

Poziotinib is an Orally Active and Irreversible pan-HER Inhibitor

2021-01-15 Edward Jenner

The HER protein is a transmembrane tyrosine kinase receptor and a member of the epidermal growth factor receptors (EGFRs) family.…

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Posted in: Cancer Immunotherapy Filed under: Antitumor, Apoptosis, EGFR, HER, SNU216

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Recent Posts

  • GSK3036656 is an orally active inhibitor of M. tuberculosis leucyl-tRNA synthetase 2022-06-25
  • Toceranib (SU11654) is an Orally Active RTK Inhibitor 2022-06-23
  • ALK4290 (AKST4290) is an Orally Active CCR3 Inhibitor 2022-06-21

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