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Tag: Histamine

S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor

2021-02-24 Edward Jenner

Histamine is an important neurotransmitter exerting its actions via four classes of molecularly and/or pharmacologically well-defined receptors. They differ in…

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Posted in: Neurological Disease Filed under: BDNF, H3, Histamine, VEGF

A-987306 is a Potent and Orally Active Histamine H4 Antagonist

2020-09-08 Edward Jenner

Histamine exhibits its functions through four known G-protein coupled receptors, the H1, H2, H3, and H4 receptors. Some histamine receptor…

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Posted in: Inflammation Filed under: Histamine, Hyperalgesia, Peritonitis

PF-03654764 is a Selective Histamine H3 Receptor Antagonist

2020-07-29 Edward Jenner

The symptoms of Allergic rhinitis are rhinorrhea, sneezing, nasal pruritus, congestion, and aggravation of comorbid asthma. Histamine can interact with…

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Posted in: Allergy, Rhinitis Filed under: H3, Histamine

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