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Autoimmune diseases

Deucravacitinib is an Orally Active TYK2 Allosteric Inhibitor for Autoimmune Diseases Research

Edward Jenner 2023-04-11

Tyrosine kinase 2 (TYK2) is a member of the JAK kinase family. Besides, it regulates signal transduction downstream of the IL-23/IL-12 pathway and the type I interferon family receptor, pairing…

Cancer Immunotherapy Immunotherapy Innate Immune

TAK-676 is a STING Agonist and Triggers the STING Signaling Pathway Activation

Edward Jenner 2022-09-03

Stimulator of interferon genes (STING), an integral ER-membrane protein, is a protein that in humans is encoded by the STING1 gene. STING plays an important role in innate immunity. It…

Autoimmune Disorders Inflammation Innate Immune

C-178 is a Covalent Small-Molecule Inhibitor of STING

Edward Jenner 2019-09-26

In the previous blog, I have introduced C-176 as a strong and covalent mouse STING inhibitor. Today, I’d like to introduce another STINF inhibitor C-178 in the same article. STING,…

Inflammation Rheumatoid Arthritis

PS372424 is a Specific Agonist for The Human CXCR3

Edward Jenner 2019-07-11

Chemokines are low-molecular weight proteins that mediate the migration of leucocytes. Crucially, chemokines exert their effects by binding to specific GPCRs expressed on the leucocyte surface. Of these, the chemokine…

Innate Immune

MRT67307 is a Dual Inhibitor of the IKKε and TBK-1

Edward Jenner 2019-07-02

IKK {IκB kinase} family plays a indispensable role in innate immunity by inducing NF-κB- and IRF -dependent gene transcription programmes required for the production of pro-inflammatory cytokines and IFNs. A…

Inflammation

NG25, a Dual Inhibitor of TAK1 and MAP4K2, Suppresses Production of IFNα

Edward Jenner 2019-06-24

TAK1 is also called Mitogen-activated protein kinase kinase kinase 7 (MAP3K7). It belongs to the serine/threonine protein kinase family. The kinase regulates cell death, and its activation is through a…

Auto-Inflammatory Inflammation Innate Immune

C-176 is a Covalent Small Molecule Inhibitor of STING

Edward Jenner 2019-04-05

The abnormal activation of innate immune pathways partispate in the progress of various diseases. Unfortunately, the development of drugs specifically targeted molecules with interest and potential still remains challenging. A…

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  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
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  • Doravirine is a HIV-1 Inhibitor for Infection Research

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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

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