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Tag: Interferon

C-178 is a Covalent Small-Molecule Inhibitor of STING

2019-09-26 Edward Jenner

In the previous blog, I have introduced C-176 as a strong and covalent mouse STING inhibitor. Today, I’d like to…

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Posted in: Autoimmune Disorders, Inflammation, Innate Immune Filed under: Interferon, STING

PS372424 is a Specific Agonist for The Human CXCR3

2019-07-11 Edward Jenner

Chemokines are low-molecular weight proteins that mediate the migration of leucocytes. Crucially, chemokines exert their effects by binding to specific…

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Posted in: Inflammation, Rheumatoid Arthritis Filed under: Anti-Inflammatory, CXCR3, Interferon

MRT67307 is a Dual Inhibitor of the IKKε and TBK-1

2019-07-02 Edward Jenner

IKK {IκB [inhibitor of NF-κB (nuclear factor κB)] kinase} family plays a indispensable role in innate immunity by inducing NF-κB-…

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Posted in: Innate Immune Filed under: IKK, Interferon, TBK

NG25, a Dual Inhibitor of TAK1 and MAP4K2, Suppresses Production of IFNα

2019-06-24 Edward Jenner

TAK1 is also called Mitogen-activated protein kinase kinase kinase 7 (MAP3K7). It belongs to the serine/threonine protein kinase family. The…

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Posted in: Inflammation Filed under: Cytokine, Interferon, Interleukin

C-176 is a Covalent Small Molecule Inhibitor of STING

2019-04-05 Edward Jenner

The abnormal activation of innate immune pathways partispate in the progress of various diseases. Unfortunately, the development of drugs specifically…

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Posted in: Auto-Inflammatory, Inflammation, Innate Immune Filed under: Auto-inflammatory, Interferon, STING

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Anti-Inflammatory Anti-Tumor Antibacterial Antimalarial Antitumor Antiviral Apoptosis Autophagy Breast Cancer Btk Chemokines COPD COX Cytokine EGFR ER Stress HBV HCV HDAC HIV IFN IL-6 IL-17 Infection Integrin Interferon Interleukin Leukemia Low Toxicity Multidrug Resistance Necroptosis NF-κB p38 MAPK PI3K PPI Proteasome RIPK STAT STING T Cell Th17 TLR TNF TNF-α α4β1
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