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Tag: Leukemia

NMS-E973 is a Selective and BBB-Penetrated HSP90 Inhibitor

2020-11-17 Edward Jenner

Hsp90 is a molecular chaperone, it is essential for the conformational stability and activity of many key oncogenic proteins. These…

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Posted in: Cancer Immunology Filed under: BT-474, CAL-51, DU-4475, HCC1419, HCC1954, HSP90, Leukemia

BMS-906024 is an Orally Active γ-Secretase and Notch Inhibitor

2020-09-23 Edward Jenner

Gamma secretase (γ-Secretase) is a kind of multi-subunit protease complex, which is an indispensable membrane protein. Specifically, γ-Secretase cleaves one-way…

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Posted in: Cancer Immunology Filed under: Leukemia, Lung Adenocarcinoma, Notch, Solid Tumor, γ-Secretase

MI-3454 is an Orally Active Menin-MLL1 Interaction Inhibitor

2020-06-24 Edward Jenner

The protein-protein interaction between menin and MLL fusion proteins plays a critical role in the pathogenesis of MLL leukemia. The…

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Posted in: Cancer Immunology Filed under: Leukemia, Menin, MLL1

A-205804 is a Selective Inhibitor of E-selectin and ICAM-1

2020-04-30 Edward Jenner

Integrins are transmembrane receptors that facilitate cell-extracellular matrix (ECM) adhesion. The presence of integrins allows rapid and flexible responses to…

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Posted in: Cancer Immunology Filed under: E-selectin, Leukemia

TEI-9647, a Vitamin D antagonist, Inhibits Osteoclast Formation

2020-03-05 Edward Jenner

The vitamin D receptor (VDR) is a member of the nuclear receptor family of transcription factors. 1α,25(OH)2D3 is to mediate biological…

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Posted in: Immunology Filed under: Leukemia, Osteoclast, VDR

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