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HIV Viral Immunology

TMC310911 is a Potent and Orally Active HIV-1 Protease Inhibitor

Edward Jenner 2020-04-28

The human immunodeficiency viruses (HIV) are two species of Lentivirus that infect humans. It causes acquired immunodeficiency syndrome (AIDS). Besides, AIDS is a condition in which progressive failure of the…

Cancer Immunology

ZX-29, a Selective ALK Inhibitor, Induces Apoptosis via ER Stress

Edward Jenner 2020-04-16

Anaplastic lymphoma kinase (ALK) is a member of the insulin receptor superfamily. Specifically, the fusion form can activate ALK, and ALK is continuously activated. Besides, the abnormal activation of ALK abnormally…

Bacterial Infection

PK150 is an Orally Active Antibacterial Compound

Edward Jenner 2020-02-18

The current treatment of bacterial infections is challenged by a dramatic increase of multidrug-resistant (MDR) strains. In addition to Gram-negative MDR pathogens cause infection, Gram-positive pathogens, such as Staphylococcus aureus,…

Bacterial Inflammation

SPR741, an Anti-biotic Potentiator, Inhibits Multidrug-Resistant Gram-negative Bacteria

Edward Jenner 2019-12-16

SPR741, an antibiotic adjuvant that can permeabilize the Gram-negative membrane. In this article, we will briefly introduce this compound in vitro and in vivo. SPR741 lacks significant antibacterial activity as…

Malaria Parasite

TCMDC-135051, a Highly Selective PfCLK3 Inhibitor, Has Potential to Treat Malaria

Edward Jenner 2019-09-20

PfCLK3 is a protein kinase essential for maintaining the asexual blood stage of both P. falciparum and P. berghei.  In mammalian cells, the CLK protein kinase family and the closely related SRPK family…

Bacterial Tuberculosis

VXc-​486, a Gyrase B Inhibitor, Has Potential to Treat Tuberculosis

Edward Jenner 2019-09-19

Tuberculosis (TB) is an important infectious disease threat worldwide. HIV coinfection/immunosuppression and widespread drug resistance contributes to the challenge of controlling TB. TB resulted from Mycobacterium tuberculosis. It is a…

Bacterial

An Efflux Pump AcrB and MexB Inhibitor D13-9001

Edward Jenner 2019-05-16

Multidrug resistance (MDR) provokes obstruction in disease control by intensifying the possibility of spreading of resistant pathogens. It declines efficacy of treatment and, hence, resulting in prolonged time of infection…

Recent Posts

  • Mirikizumab is a Humanized IgG4 mAb for Ulcerative Colitis Research
  • Grazoprevir is a Hepatitis C virus NS3/4A Protease Inhibitor for Infection Research
  • Efbemalenograstim alfa is a Recombinant Fusion Protein for Neutropenia Research
  • Remibrutinib is an Orally Active BTK Inhibitor for Chronic Urticaria Research
  • Taurolidine is a Broad-spectrum Antimicrobial for Central Venous Catheter-Related Infections Research

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You Missed

Inflammation Ulcerative Colitis

Mirikizumab is a Humanized IgG4 mAb for Ulcerative Colitis Research

Hepatitis Hepatitis C Virus

Grazoprevir is a Hepatitis C virus NS3/4A Protease Inhibitor for Infection Research

Breast cancer Infection

Efbemalenograstim alfa is a Recombinant Fusion Protein for Neutropenia Research

Cancer Chronic Urticaria Inflammatory Uncategorized

Remibrutinib is an Orally Active BTK Inhibitor for Chronic Urticaria Research

Immune System Research

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