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Tag: PI3K

IHMT-PI3Kδ-372 is a Potent and Selective PI3Kδ Inhibitor

2021-01-06 Edward Jenner

PI3Kδ belongs to the class I Phosphoinositide 3-kinases (PI3Ks). PI3Kδ plays a critical role in chronic obstructive pulmonary disease (COPD).…

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Posted in: Chronic Obstructive Pulmonary Disease, Inflammation Filed under: AKT, COPD, PI3K, PI3Kδ

MSC2360844 is an Orally Active and Selective PI3Kδ Inhibitor

2020-11-07 Edward Jenner

SLE is a complex autoimmune inflammatory disease that affects multiple organs with unpredictable flares. Autoantibody/antigen immune-complexes in turn can activate…

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Posted in: Autoimmune Disorders, Lupus Nephritis Filed under: IFNα, PI3K, SLE, TLR

AQX-435 is a Potent SHIP1 Activator and an Apoptosis Inducer

2020-10-28 Edward Jenner

PI3Ks are key drivers of the survival and growth of normal B cells. PI3K catalyzes the phosphorylation of PI(4,5)P2 to…

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Posted in: Cancer Immunology Filed under: Apoptosis, Lymphoma, PI3K, SHIP1

GS-9901, an Orally Active PI3Kδ Inhibitor, Has Potential to Treat Rheumatoid Arthritis

2019-07-24 Edward Jenner

Phosphoinositide 3-kinase (PI3K) plays an indispensable role in the signal transduction of numerous cellular functions via the formation of the…

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Posted in: Rheumatoid Arthritis Filed under: Anti-Inflammatory, PI3K

LAS191954 is an Orally Active PI3Kδ Inhibitor

2019-07-23 Edward Jenner

The phosphatidylinositol-3-kinase (PI3K) signal transduction pathway plays an indispensable role in different cellular processes involving metabolism, proliferation, differentiation or activation.…

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Posted in: Inflammation Filed under: Anti-Inflammatory, PI3K

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