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Tag: Stroke

GKT136901 is a Selective and Orally Active Inhibitor of NADPH Oxidase (NOX1/4)

2020-10-24 Edward Jenner

NADPH oxidases (NOX), catalyzing the reduction of molecular oxygen to form the superoxide radical anion (O₂⁻) and hydrogen peroxide (H₂O₂).…

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Posted in: Inflammation Filed under: NADPH Oxidase, Nox, Stroke, Type 2 Diabetes

RP101075 is a Potent and Orally Active S1PR Agonist

2020-07-25 Edward Jenner

Sphingosine-1-phosphate (S1P) is a ligand for G-protein-coupled receptors, it is responsible for some cell-intrinsic and extrinsic activities. RPC1063 is a…

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Posted in: Immunology Filed under: ICH, S1PR, Safe, Stroke

IOX4 is a Highly Selective PHD2 Inhibitor

2019-09-17 Edward Jenner

Prolyl hydroxylases (PHDs) target hypoxia-inducible factor-1α (HIF-1α) for degradation. Hypoxia inactivates PHDs, causing accumulation of HIF-1α. In turn, HIF-1 further…

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Posted in: Cancer Immunology, Neurological Disease Filed under: HIF, PHD, Stroke

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