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Immune System Research

Up to date immunology information.

Cyclocurcumin is a Potent p38α Inhibitor for Rheumatoid Arthritis Research

2023-05-31 Edward Jenner

p38 mitogen-activated protein kinase (MAPK) plays a key role in cellular response, proliferation, survival, cell cycle and cancer migration. Moreover, the…

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Posted in: Arthritis Filed under: Anti-vasoconstrictive, Antirheumatic, p38α, rheumatoid arthritis

Efipladib is an Orally Active cPLA2α Inhibitor for Inflammation Research

2023-05-30 Edward Jenner

cPLA2α is an intracellular calcium dependent PLA2. It is expressed in a wide variety of tissues and cells. Firstly, cPLA2α…

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Posted in: Inflammation Filed under: COX-2, cPLA2α, Efipladib, Inflammation, Oral, PLA2

Fezolinetant is a NK3R Antagonist for Menopausal Hot Flushes Research

2023-05-29 Edward Jenner

Neurokinin 3 receptor (NK3R) is the most selective of the tachykinin receptors, with highly preferential binding and activation by its…

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Posted in: Endocrinology, Hot flushes Filed under: Fezolinetant, Hot flushes, NK3R

TYA-018 is an Orally Active HDAC6 Inhibitor for Cardiovascular Disease Research

2023-05-26 Edward Jenner

Dilated cardiomyopathy (DCM) is a form of heart muscle weakness. Firstly, it shows the reduction of cardiac output, as well…

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Posted in: Cardiovascular, Dilated cardiomyopathy disease Filed under: cardiovascular disease, Dilated cardiomyopathy disease, HDAC, Oral, TYA-018

CP-465022 is a Noncompetitive AMPA Receptor Antagonist for Neurological Disease Research

2023-05-25 Edward Jenner

The α-amino-3-hydroxy-5-methyl-4-isoxazolopropionic acid receptor (AMPA receptor) is an ionic glutamate (iGluR) transmembrane receptor. Specifically, it can mediate the rapid synaptic…

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Posted in: Neurological Disease Filed under: AMPA, Anticonvulsant, CP-465022, NMDA

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