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Immune System Research

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KSC-34 is a Site-Selective Inhibitor of PDIA1

2021-02-17 Edward Jenner

Proper folding of nascent proteins in the cell is accelerated by chaperones. They serve to stabilize protein domains and overall…

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Posted in: Immunology Filed under: PDI, PDIA1

NGB 2904 is an Orally Active and Brain-Penetrated Antagonist of Dopamine D3 Receptor

2021-02-16 Edward Jenner

Drug abuse is a serious health problem in many areas of the world. There are no widely effective medications available…

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Posted in: Neurological Disease Filed under: 5-HT, Cocaine, D3 Receptor, Dopamine

L-368,899 is a Selective and Orally Active Oxytocin Receptor Antagonist

2021-02-13 Edward Jenner

L-368,899 is a potent, orally bioavailable, non-peptide oxytocin receptor antagonist. L-368,899 shows IC50s of 8.9 nM and 26 nM for…

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Posted in: Endocrinology Filed under: Oxytocin, Vasopressin

Sisunatovir is an Orally Available Inhibitor of the RSV Fusion (RSV-F) Protein

2021-02-11 Edward Jenner

Respiratory syncytial virus (RSV) is an enveloped, single-stranded, negative-sense RNA virus. It belongs to the Pneumovirinae subfamily of Paramyxoviridae.  Furthermore, this kind of…

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Posted in: Respiratory Infection Filed under: Respiratory Syncytial Viral, RSV, RSV-F

UCB-9260 Inhibits TNF Signalling by Stabilising an Asymmetric form of the Trimer

2021-02-10 Edward Jenner

Tumor necrosis factor (TNF) is a cytokine belonging to a family of trimeric proteins. This factor acts as a key…

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Posted in: Arthritis, Collagen-Induced Arthritis Filed under: CAIA, TNF

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  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24
  • FSCPX is a Selective Irreversible Antagonist of A1AR 2021-02-23

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