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Immune System Research
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Tag: 5-HT

SCH-23390 is a Selective Dopamine D1-Like Receptor Antagonist

2021-12-28 Edward Jenner

Dopamine Receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Abnormal…

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Posted in: Neurological Disease Filed under: 5-HT, Dopamine, GIRK, Inflammasome, NLRP3, Potassium Channel

FAUC 346 is a Highly Selective D3 Partial Agonist

2021-06-17 Edward Jenner

Dopamine receptors are classified into the Gs-coupled D1-like (D1 and D5) and Gi/o-coupled D2-like (D2, D3, and D4) receptor subtypes.…

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Posted in: Neurological Disease Filed under: 5-HT, Cocaine, D3, Dopamine

SB-203186 is a Selective and Competitive 5-HT4 Antagonist

2021-05-22 Edward Jenner

5-HT receptors are a group of G protein-coupled receptors and ligand-gated ion channels in the central nervous system and peripheral…

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Posted in: Cardiovascular Filed under: 5-HT, Tachycardia

SEP-363856 is an Orally Active Psychotropic Agent with a non-D2/5-HT2A Action

2021-04-27 Edward Jenner

Antipsychotics are a class of medication for managing psychosis, principally in schizophreniabut also in a range of other psychotic disorders.…

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Posted in: Parkinson’s, Schizophrenia Filed under: 5-HT, Antipsychotic, TAAR1

NGB 2904 is an Orally Active and Brain-Penetrated Antagonist of Dopamine D3 Receptor

2021-02-16 Edward Jenner

Drug abuse is a serious health problem in many areas of the world. There are no widely effective medications available…

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Posted in: Neurological Disease Filed under: 5-HT, Cocaine, D3 Receptor, Dopamine

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