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Tag: CCR

TAK-779 is an Antagonist of CCR5 and CXCR3, with Anti-HIV-1 Effect

2019-08-12 Edward Jenner

Nowadays, people are no strangers to AIDS. It is a kind of infectious disease caused by HIV. The latter primarily…

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Posted in: Arthritis, Asthma, Autoimmune Disorders, Viral Immunology Filed under: Anti-Inflammatory, Anti-Tumor, CCR, HIV

BX471 is a Potent and Selective CCR1 Antagonist

2019-07-04 Edward Jenner

Renal ischemia/reperfusion injury (IR) is a major clinical problem found in shock, renal transplantation and other clinical settings. Neutrophils and…

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Posted in: Autoimmune Disorders, Inflammation Filed under: Anti-Inflammatory, CCR, Chemokines

RS 504393 is a Selective CCR2 Chemokine Receptor Antagonist

2019-07-03 Edward Jenner

Monocyte chemoattracant-1 (MCP-1) stimulates leukocyte chemotaxis to inflammatory sites, such as rheumatoid arthritis, atherosclerosis, and asthma, by use of the…

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Posted in: Allergy, Fibrosis, Inflammation Filed under: CCR, Chemokines

AZ084, a CCR8 Antagonist, Inhibits Dendritic Cell, T Cell and Eosinophil Migration

2019-06-08 Edward Jenner

The prevalence of asthma and the associated cost burden for the health care system is high. The chemokine receptor Chemokine…

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Posted in: Asthma, Respiratory Infection Filed under: Anti-Inflammatory, CCR

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Recent Posts

  • WEHI-9625, a VDAC2:BAK Interaction Enhancer, Blocks mBAK-Mediated Apoptosis 2021-02-25
  • S 38093 is a Brain-Penetrant and Orally Active Antagonist of H3 Receptor 2021-02-24
  • FSCPX is a Selective Irreversible Antagonist of A1AR 2021-02-23

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