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Cancer

SLMP53-2 is a Mutant p53 Reactivator for Cancer Research

Edward Jenner 2023-07-14

p53 (Tumor protein P53; cellular tumor antigen p53; transformation-related protein 53 (TRP53)) is a regulatory protein. The p53 proteins are crucial in vertebrates, where they prevent cancer formation. As such,…

Cancer Immunology Infection

Tunicamycin Inhibits N-linked Glycosylation, GlcNAc Phosphotransferase and Induces ER Stress

Edward Jenner 2021-08-28

N-linked glycosylation (NLG) is the attachment of an oligosaccharide and a nitrogen atom (the amide nitrogen of an asparagine (Asn) residue of a protein) in a process called N-glycosylation. NLG…

Autoimmune Disorders Inflammation

GSK-J4 is a Dual Inhibitor of H3K27me3/me2-Demethylases JMJD3/KDM6B and UTX/KDM6A

Edward Jenner 2021-02-18

H3K27me3 is an epigenetic modification of DNA packaging protein histone H3. Specifically, it is a marker for the trimethylation of lysine 27 on histone H3 protein. Besides, H3K27me3 is relevant…

Cancer Immunology

PACMA 31 is an Irreversible and Orally Active Protein Disulfide Isomerase (PDI) Inhibitor

Edward Jenner 2020-12-08

Ovarian cancer is one of the leading causes of death in women with gynecological cancers in the United States. About 70% of ovarian cancer cases are diagnosed at a late…

Neuroimmunology

MK-28 is a Potent and Selective PERK Activator

Edward Jenner 2020-10-15

Protein kinase R (PKR)-like endoplasmic reticulum kinase (PERK) is an endoplasmic reticulum-associated stress sensor protein. PERK phosphorylates eukaryotic initiation factor 2α (eIF2α) to induce translation attenuation in response to ER…

Cancer Immunology

ZX-29, a Selective ALK Inhibitor, Induces Apoptosis via ER Stress

Edward Jenner 2020-04-16

Anaplastic lymphoma kinase (ALK) is a member of the insulin receptor superfamily. Specifically, the fusion form can activate ALK, and ALK is continuously activated. Besides, the abnormal activation of ALK abnormally…

Fibrosis Pulmonary Fibrosis

KIRA-7 is an Allosteric IRE1α Kinase/Rnase Inhibitor

Edward Jenner 2020-02-25

Idiopathic pulmonary fibrosis (IPF) is a disease of progressive fibrosis and respiratory failure. Endoplasmic reticulum stress (ER stress) implicates in the pathogenesis of idiopathic pulmonary fibrosis. ER stress activates a…

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  • PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH
  • Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research
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You Missed

Pulmonary Arterial Hypertension (PAH)

PRX-08066 is an orally active 5-HT2BR Antagonist with Vasodilation Effect for PAH

Cancer Immune Metabolic Disease

Apocynin is a NADPH oxidase (NOX) Inhibitor for Metabolic and Inflammation Research

Uncategorized

Xylometazoline is an α-adrenergic Receptor Agonist for Nose Stuffiness Research

NASH obesity

Elafibranor is a PPARα/δ Agonist for Metabolic Disease Research

Immune System Research

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